Target Details
| UniProt AC | P17301 |
|---|---|
| Gene Symbol | ITGA2 |
| Protein Name | Integrin alpha-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00092 (VWA) |
Summary
- Multi-target molecules 65
- Clinical molecules 0
- Avg pChEMBL 7.24
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phagosome
- Platelet activation
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Small cell lung cancer
- Virion - Rotavirus
Associated Diseases (2)
Active Molecules (65)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBEWYOLFNVQHDU
|
6.5 | IC50 | 3 | — | |
JXCMMMJBHLWVLH
|
6.5 | IC50 | 3 | — | |
CNVZYIOAIFJZCD
|
6.4 | IC50 | 2 | — | |
MXVNNRPZXJVWDK
|
6.3 | IC50 | 2 | — | |
DVUDJTXPOUYIBT
|
6.3 | IC50 | 2 | — | |
NSAHPDSQIRNDGO
|
6.2 | IC50 | 2 | — | |
GSBDJNSXYKUYNP
|
6.2 | IC50 | 2 | — | |
FBEWYOLFNVQHDU
|
6.2 | IC50 | 3 | — | |
MVOPMYAHCQTVSN
|
6.1 | IC50 | 2 | — | |
VOZWZDMFSQVZQP
|
6.1 | IC50 | 2 | — | |
CTVYHQCWCNHILX
|
6.1 | IC50 | 2 | — | |
DPBYUKDFQVKXHU
|
6.1 | IC50 | 2 | — | |
TUEFPOMKBBGSEI
|
6.1 | IC50 | 2 | — | |
XXVHVXVVXGOJQZ
|
6.0 | IC50 | 2 | — | |
NLUDZQOAPUIKSG
|
6.0 | IC50 | 2 | — |