Target Details
| UniProt AC | P16591 |
|---|---|
| Gene Symbol | FER |
| Protein Name | Tyrosine-protein kinase Fer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00611 (FCH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 164
- Clinical molecules 21
- Avg pChEMBL 6.85
KEGG Pathways (1)
Active Molecules (164)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XKZINYYXWJEYEL
|
6.5 | Ki | 37 | — | |
ZKHDDJKHTPLPOQ
|
6.5 | Ki | 62 | — | |
MGGBYMDAPCCKCT
|
6.4 | Kd | 23 | — | |
FLBNLJLONKAPLR
|
6.4 | Kd | 31 | — | |
BSFNGHCTZDCQBF
|
6.4 | Ki | 93 | — | |
CLEGDJQQHUTCOW
|
6.4 | Ki | 43 | — | |
MASJMHFQMYAPJR
|
6.4 | Ki | 41 | — | |
NRSGWEVTVGZDFC
|
6.4 | Ki | 50 | — | |
RYAVJHIPOWNWDE
|
6.4 | Ki | 38 | — | |
PBCZSGKMGDDXIJ
|
6.4 | Kd | 68 | Yes | |
KOZFSFOOLUUIGY
|
6.3 | Kd | 88 | Yes | |
UBPYILGKFZZVDX
|
6.3 | Kd | 130 | Yes | |
IFQICUARAXVEIQ
|
6.3 | Ki | 18 | — | |
LGHBDVLAHHANMX
|
6.3 | Ki | 53 | — | |
MPVGZUGXCQEXTM
|
6.3 | Ki | 61 | Yes | |
OUJZYQBEFNDJQN
|
6.3 | Ki | 71 | — | |
UUWNXFJBBYAMDT
|
6.3 | Ki | 46 | — | |
XPPLYAKZGXYPOZ
|
6.3 | Ki | 6 | — | |
ZGDSBEUMPIMXBM
|
6.3 | Ki | 42 | — | |
JWNPDZNEKVCWMY
|
6.3 | Kd | 57 | Yes | |
PDOQBOJDRPLBQU
|
6.3 | Kd | 21 | — | |
FCNPQYHKUYSELK
|
6.2 | IC50 | 8 | — | |
WKDACQVEJIVHMZ
|
6.2 | Kd | 46 | — | |
ODPGGGTTYSGTGO
|
6.2 | Kd | 153 | — | |
HHSVICUMCOBRPT
|
6.2 | Ki | 33 | — | |
KJVWCDAPVMWKLJ
|
6.2 | Ki | 20 | — | |
PPCNMZPSQZFFGM
|
6.2 | Ki | 8 | — | |
VUHZDNOPEVGHEO
|
6.2 | Ki | 29 | — | |
SLEWGGZPOQNVSU
|
6.2 | Kd | 22 | — | |
XKFTZKGMDDZMJI
|
6.2 | Kd | 64 | Yes | |
ACNCCUVYXQGPKZ
|
6.1 | Ki | 31 | — | |
AYCPARAPKDAOEN
|
6.1 | Kd | 73 | — | |
BHSOPYVVEZFHDB
|
6.1 | Ki | 25 | Yes | |
DKSNLQYRZJKYOC
|
6.1 | Ki | 51 | — | |
LQVXSNNAFNGRAH
|
6.1 | Kd | 33 | Yes | |
MULNSLQVKKUPJN
|
6.1 | Ki | 41 | — | |
ORRHVRJUSPCILV
|
6.1 | Ki | 16 | — | |
QXKKPVVOOWBLND
|
6.1 | Ki | 8 | — | |
SBFPHSVZEXSHTL
|
6.1 | Ki | 62 | — | |
XJSFDMGICAWQFS
|
6.1 | Ki | 60 | — | |
YDOPLCNFRXOHCC
|
6.1 | Ki | 28 | — | |
YLCFOHVAOBLAIK
|
6.1 | IC50 | 14 | — | |
ZLVOTRRGLSDLPF
|
6.1 | Ki | 36 | — | |
MZDKLVOWGIOKTN
|
6.1 | Kd | 80 | — | |
DKNUPRMJNUQNHR
|
6.0 | Kd | 33 | — | |
ADMFLILDQJSEIK
|
6.0 | Ki | 72 | — | |
AIQDZMUPVYDVLB
|
6.0 | Ki | 48 | — | |
BPNUQXPIQBZCMR
|
6.0 | Ki | 60 | — | |
CXBBWVXSZINRCS
|
6.0 | Ki | 41 | — | |
DSSRVQAIWBZWON
|
6.0 | Ki | 9 | — |