Target Details
| UniProt AC | P16591 |
|---|---|
| Gene Symbol | FER |
| Protein Name | Tyrosine-protein kinase Fer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00611 (FCH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 164
- Clinical molecules 21
- Avg pChEMBL 6.85
KEGG Pathways (1)
Active Molecules (164)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HEUSUIRCBWROMH
|
7.1 | Ki | 64 | — | |
NLUPJKQOKWBWFC
|
7.1 | Ki | 69 | — | |
SMPGEBOIKULBCT
|
7.1 | IC50 | 15 | — | |
IAYGCINLNONXHY
|
7.1 | Kd | 50 | — | |
LAJAFFLJAJMYLK
|
7.1 | IC50 | 17 | — | |
PCQMERRARZKTPW
|
7.0 | Ki | 68 | — | |
ZLHFILGSQDJULK
|
7.0 | Ki | 37 | Yes | |
RYYNGWLOYLRZLK
|
7.0 | Kd | 45 | — | |
ALKJNCZNEOTEMP
|
7.0 | Kd | 55 | — | |
ISPBCAXOSOLFME
|
7.0 | Kd | 11 | — | |
CXQHYVUVSFXTMY
|
6.9 | Kd | 154 | — | |
GUBJNPWVIUFSTR
|
6.9 | Kd | 103 | — | |
IJRBJCMLWLFMIN
|
6.9 | Ki | 17 | — | |
IZAVTOABECKIDH
|
6.9 | Ki | 20 | — | |
OADRBDVURCEKRP
|
6.9 | Ki | 44 | — | |
UOVCGJXDGOGOCZ
|
6.9 | Ki | 59 | — | |
XFWUTMHVDGPWLH
|
6.9 | Ki | 75 | — | |
XKFTZKGMDDZMJI
|
6.9 | Ki | 56 | — | |
NHHQJBCNYHBUSI
|
6.9 | Kd | 220 | — | |
AUDNGNGLLRZLDR
|
6.8 | Ki | 33 | — | |
CNTCGRJDUJEUDG
|
6.8 | Ki | 37 | — | |
GDYZFFBMSBDTAA
|
6.8 | Ki | 60 | — | |
NWAUBAGBGOPJLF
|
6.8 | Ki | 51 | Yes | |
PUPCRRRSBUYJAD
|
6.8 | Ki | 44 | Yes | |
DLWMVUDMPMKGEE
|
6.7 | Ki | 24 | — | |
FDVSOQRNTAPCHB
|
6.7 | Ki | 40 | — | |
FUMCKNCUEAQHCV
|
6.7 | Ki | 103 | — | |
IOBVCHJTLVPPBR
|
6.7 | Ki | 39 | — | |
KOHNRDPXFDZZJF
|
6.7 | Ki | 31 | — | |
VERWOWGGCGHDQE
|
6.7 | Kd | 23 | — | |
OYKPWSZSBLRRPL
|
6.6 | IC50 | 11 | — | |
DBXGGXLBTWZXBB
|
6.6 | Ki | 39 | — | |
NRGYZNJPCGRCLV
|
6.6 | Ki | 52 | — | |
OWFXKTOLFUQPDJ
|
6.6 | Ki | 36 | — | |
PTVPBWWDGZSEAF
|
6.6 | Ki | 63 | — | |
UOOZSMNSBYVUGZ
|
6.6 | Ki | 32 | — | |
WVUNYSQLFKLYNI
|
6.6 | Kd | 46 | Yes | |
XCHWBXBDZRJVDP
|
6.6 | Ki | 51 | — | |
ZGZVRPRSFXRGCF
|
6.6 | Ki | 76 | — | |
KTEIFNKAUNYNJU
|
6.6 | Kd | 114 | — | |
WVXNSAVVKYZVOE
|
6.6 | IC50 | 92 | — | |
OOMBFNDWQIGHEK
|
6.5 | Kd | 22 | — | |
LOLPPWBBNUVNQZ
|
6.5 | Kd | 97 | Yes | |
BLQYVHBZHAISJM
|
6.5 | Ki | 54 | — | |
CZQVOIDVDAVDFW
|
6.5 | Ki | 18 | — | |
LVECPYVAIBNSRV
|
6.5 | Ki | 33 | — | |
MTCHQDWUHQADSY
|
6.5 | Ki | 29 | — | |
OAVGBZOFDPFGPJ
|
6.5 | Ki | 42 | Yes | |
UDFDIIVNIYWXDM
|
6.5 | Ki | 74 | — | |
WUWDLXZGHZSWQZ
|
6.5 | Ki | 41 | — |