Target Details
| UniProt AC | P16591 |
|---|---|
| Gene Symbol | FER |
| Protein Name | Tyrosine-protein kinase Fer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00611 (FCH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 164
- Clinical molecules 21
- Avg pChEMBL 6.85
KEGG Pathways (1)
Active Molecules (164)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AILRADAXUVEEIR
|
8.9 | IC50 | 75 | — | |
LVLFSSZNAIKYCD
|
8.9 | IC50 | 19 | — | |
QQWUGDVOUVUTOY
|
8.8 | Kd | 231 | Yes | |
WHVFDYQCAMPLMS
|
8.8 | Ki | 20 | Yes | |
HKSZLNNOFSGOKW
|
8.7 | IC50 | 408 | — | |
DIXMBHMNEHPFCX
|
8.7 | IC50 | 12 | — | |
GDRLJBDXWDATLA
|
8.7 | IC50 | 13 | — | |
HKSZLNNOFSGOKW
|
8.5 | Ki | 118 | — | |
JZTOUVBEZONDKA
|
8.5 | Ki | 80 | — | |
RYYNGWLOYLRZLK
|
8.5 | Ki | 104 | — | |
IIXWYSCJSQVBQM
|
8.5 | IC50 | 18 | — | |
VXYZCOCRVAQWBG
|
8.5 | IC50 | 15 | — | |
HAYYBYPASCDWEQ
|
8.3 | Ki | 47 | — | |
ULMCFLZUGRSEQA
|
8.2 | Ki | 17 | — | |
MWKSRKSEWLRPBL
|
8.1 | Kd | 1075 | — | |
HZTYDQRUAWIZRE
|
8.0 | Kd | 40 | Yes | |
LYNBNVBMAGDJRW
|
8.0 | Ki | 81 | — | |
UYJNQQDJUOUFQJ
|
8.0 | Ki | 68 | — | |
ZCCPLJOKGAACRT
|
7.9 | Kd | 599 | — | |
MOSKATHMXWSZTQ
|
7.9 | IC50 | 16 | Yes | |
VKBFHTIUXUCYRQ
|
7.8 | Ki | 66 | — | |
MHCPAORAYMTGCZ
|
7.7 | Ki | 37 | — | |
MVJMMLFMPWITEJ
|
7.7 | Ki | 110 | — | |
XHORJSJFHVABEA
|
7.7 | Ki | 49 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
NHFDRBXTEDBWCZ
|
7.6 | Ki | 41 | — | |
XBYVOPRDASFDMY
|
7.6 | Ki | 42 | — | |
NXSJMRCTGYTSTK
|
7.6 | Kd | 200 | — | |
UIARLYUEJFELEN
|
7.5 | Kd | 289 | Yes | |
OSVUGUHRKMMBSE
|
7.5 | Kd | 170 | — | |
GCBJDOWIQHMCMR
|
7.5 | Ki | 84 | — | |
GXJSLIOOPZRPEV
|
7.5 | Ki | 34 | — | |
YMIJUBCSOKSFRU
|
7.5 | Ki | 87 | — | |
ZWVZORIKUNOTCS
|
7.5 | Ki | 69 | — | |
CTNPALGJUAXMMC
|
7.5 | Kd | 151 | — | |
KTEIFNKAUNYNJU
|
7.5 | Ki | 48 | — | |
AMHWQBGAKJESFB
|
7.4 | IC50 | 4 | — | |
SEJGTFPOEJWEGG
|
7.4 | Kd | 149 | — | |
ADLPKFFMGIJZIM
|
7.4 | Ki | 44 | — | |
DKZYXHCYPUVGAF
|
7.3 | Kd | 112 | — | |
KRIUNPBAQZGFQA
|
7.3 | Ki | 76 | — | |
WPHKIQPVPYJNAX
|
7.3 | Ki | 81 | — | |
YEHCNYAQEBQCCS
|
7.3 | Ki | 74 | — | |
MJHOMTRKVMKCNE
|
7.3 | IC50 | 12 | — | |
BIKYDWLMTPRSQL
|
7.2 | Ki | 50 | — | |
WINHZLLDWRZWRT
|
7.2 | Ki | 66 | — | |
XOOAAYRIVATZNM
|
7.2 | Ki | 55 | — | |
XZXHXSATPCNXJR
|
7.1 | Kd | 165 | Yes | |
RWNAOXLCVXJMGM
|
7.1 | IC50 | 5 | — | |
CFIBXVQLBVNOHW
|
7.1 | Ki | 64 | — |