Target Details
| UniProt AC | P16519 |
|---|---|
| Gene Symbol | PCSK2 |
| Protein Name | Neuroendocrine convertase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01483 (P_proprotein) PF00082 (Peptidase_S8) PF16470 (S8_pro-domain) |
Summary
- Multi-target molecules 9
- Clinical molecules 0
- Avg pChEMBL 8.2
Active Molecules (9)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QDGGHGYNQCXHOK
|
9.6 | Ki | 4 | — | |
UFNWIBYSOUCSGW
|
9.6 | Ki | 4 | — | |
NHBJTTGFHCHQHS
|
9.4 | Ki | 6 | — | |
PRKRCMZHFKTMTR
|
8.8 | Ki | 4 | — | |
WPZVXHODDBZCLI
|
8.8 | Ki | 4 | — | |
CLTYJDDMFQEKEL
|
7.3 | Ki | 6 | — | |
QMAXHSLPLMYIPN
|
7.3 | Ki | 6 | — | |
RARQEZVPGNQDRL
|
6.5 | Ki | 5 | — | |
YGMAIAXBJLVVLI
|
6.5 | Ki | 5 | — |