Target Details
| UniProt AC | P16473 |
|---|---|
| Gene Symbol | TSHR |
| Protein Name | Thyrotropin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF13306 (LRR_5) |
Summary
- Multi-target molecules 14
- Clinical molecules 0
- Avg pChEMBL 7.33
KEGG Pathways (6)
Associated Diseases (2)
Top Co-occurrence Targets
- FSHR 14 shared
Active Molecules (14)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IOEFWCOWBKDSQX
|
8.0 | IC50 | 2 | — | |
IOEFWCOWBKDSQX
|
8.0 | IC50 | 2 | — | |
MYYNESYILJSLRM
|
7.6 | IC50 | 2 | — | |
XEGSXAZIAWXAJO
|
7.5 | IC50 | 2 | — | |
QPOHDSYISGKVTN
|
7.5 | IC50 | 2 | — | |
VZHDZZCDHHJVAP
|
7.3 | IC50 | 2 | — | |
IMAMZGOYNNFNBX
|
7.3 | IC50 | 2 | — | |
QMPZDUZCXNFISC
|
7.2 | IC50 | 2 | — | |
BQJACMMFLPJGCR
|
7.2 | IC50 | 2 | — | |
JDELMZBOFIXWGA
|
7.2 | IC50 | 2 | — | |
PRNNNUJEBJXVGU
|
7.1 | IC50 | 2 | — | |
LOEKKSRIIAJKNW
|
7.0 | IC50 | 2 | — | |
LTNPDFQEDQPSGC
|
6.9 | IC50 | 2 | — | |
SDXOTRLCWRFJCY
|
6.7 | IC50 | 2 | — |