Target Details
| UniProt AC | P16234 |
|---|---|
| Gene Symbol | PDGFRA |
| Protein Name | Platelet-derived growth factor receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 860
- Clinical molecules 94
- Avg pChEMBL 7.24
KEGG Pathways (22)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Focal adhesion
- Gap junction
- Glioma
- Human cytomegalovirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (4)
Active Molecules (860)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ADFZKKWKESWUFY
|
7.3 | IC50 | 8 | — | |
WOSKHXYHFSIKNG
|
7.3 | IC50 | 24 | — | |
JNFPOOBKOALVEY
|
7.3 | Ki | 6 | — | |
ORYMWWSJZRCUSV
|
7.3 | IC50 | 7 | — | |
VQQRGHOPEJXFCR
|
7.3 | IC50 | 3 | — | |
AQSOVJFZYARRIS
|
7.3 | Ki | 6 | — | |
HAZVCDSGCISCHC
|
7.3 | IC50 | 3 | — | |
ICESXCDRPZKRHM
|
7.3 | IC50 | 5 | — | |
KHZNPBYKXJANSV
|
7.3 | IC50 | 4 | — | |
MHUDJGJLMGAWOB
|
7.3 | Ki | 6 | — | |
PIQCTGMSNWUMAF
|
7.3 | Kd | 137 | Yes | |
PJYLAPUQQYSUKA
|
7.3 | IC50 | 5 | — | |
FPZFOTHNFGTZRK
|
7.3 | IC50 | 2 | — | |
MUTDSMFDBHESKX
|
7.3 | IC50 | 2 | — | |
NAHZLQDLUYGRTF
|
7.3 | IC50 | 4 | — | |
FOFDIMHVKGYHRU
|
7.2 | IC50 | 2 | — | |
JPKSISIJPSXDLA
|
7.2 | IC50 | 10 | Yes | |
OYHXDIYGCSLVFT
|
7.2 | IC50 | 4 | — | |
RORITMKRNLYYLH
|
7.2 | IC50 | 2 | — | |
SZETXTFRBXNRRT
|
7.2 | IC50 | 2 | — | |
ZSOHVWILRHPULK
|
7.2 | IC50 | 3 | — | |
AOLUUEDZXBVWED
|
7.2 | IC50 | 2 | — | |
AVQNZSIEXOYAGE
|
7.2 | IC50 | 6 | — | |
GXKSGTIXGWDSGJ
|
7.2 | IC50 | 12 | Yes | |
OQBJXGADOAMRSR
|
7.2 | IC50 | 5 | — | |
UIIZAHJFDOZUIV
|
7.2 | IC50 | 3 | — | |
UKJTWBAIJVXDSM
|
7.2 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
7.2 | Kd | 85 | Yes | |
MZPQDMUNWXBKLC
|
7.2 | IC50 | 3 | — | |
OAKGNIRUXAZDQF
|
7.2 | IC50 | 2 | — | |
OAKGNIRUXAZDQF
|
7.2 | IC50 | 3 | — | |
BEFUAVPFBGOHKT
|
7.2 | IC50 | 2 | — | |
HKIJOVMUJUDWGI
|
7.2 | IC50 | 4 | — | |
MLFZJIDNGFABRH
|
7.2 | IC50 | 3 | — | |
YWTXHHRPNVQPIM
|
7.2 | IC50 | 3 | — | |
BTTQBEBOAWSMQZ
|
7.2 | IC50 | 3 | — | |
WBIIAZNRHKEMQF
|
7.2 | IC50 | 4 | — | |
WQWAOPKSXYOQPY
|
7.2 | IC50 | 3 | — | |
CYVRFHRDWQAJGA
|
7.2 | IC50 | 2 | — | |
LFKQSJNCVRGFCC
|
7.2 | IC50 | 6 | — | |
REWMPRKUAPYNBX
|
7.2 | IC50 | 2 | — | |
KVSCJEFMRSEDOZ
|
7.2 | IC50 | 2 | — | |
NXAGIDNAFCDRSJ
|
7.2 | IC50 | 2 | — | |
NZUICIGFUCOURS
|
7.2 | IC50 | 4 | — | |
QFCXANHHBCGMAS
|
7.2 | IC50 | 7 | — | |
SQHKULNLQJHPDX
|
7.2 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
7.2 | IC50 | 92 | — | |
ZJIOVLLLFWQBKA
|
7.2 | IC50 | 2 | — | |
TVLKSGDRIZGJII
|
7.1 | IC50 | 3 | — | |
DAZCBQNFGSWSQG
|
7.1 | IC50 | 8 | Yes |