Target Details
| UniProt AC | P16234 |
|---|---|
| Gene Symbol | PDGFRA |
| Protein Name | Platelet-derived growth factor receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 860
- Clinical molecules 94
- Avg pChEMBL 7.24
KEGG Pathways (22)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Focal adhesion
- Gap junction
- Glioma
- Human cytomegalovirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (4)
Active Molecules (860)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VBQLMMTYTIVERQ
|
7.5 | Ki | 6 | — | |
DIMLYBUSJYNUFT
|
7.5 | IC50 | 6 | — | |
OFLUDTFEINFEBP
|
7.5 | Ki | 6 | — | |
TWOLOZGQZKJZKJ
|
7.5 | IC50 | 7 | Yes | |
ZZYRQSFRXAHEJU
|
7.5 | Ki | 6 | — | |
AMZWYWQCAVGQIH
|
7.4 | IC50 | 3 | — | |
ARFSBNIXMVQEPO
|
7.4 | IC50 | 2 | — | |
RBARWKMXQSXULQ
|
7.4 | IC50 | 3 | — | |
RJAKZMKAAHGXTE
|
7.4 | Ki | 6 | — | |
BIVCQZJNUCQVNS
|
7.4 | IC50 | 2 | — | |
RBNNHHFJDATPRT
|
7.4 | IC50 | 2 | — | |
GBJVVSCPOBPEIT
|
7.4 | Kd | 13 | Yes | |
GNIYUURCQFKRCB
|
7.4 | IC50 | 11 | Yes | |
QYZOGCMHVIGURT
|
7.4 | Kd | 26 | Yes | |
VXNRKGFHJWQYFY
|
7.4 | Ki | 6 | — | |
BCDAHFZFGKOCPG
|
7.4 | IC50 | 4 | — | |
BLQYVHBZHAISJM
|
7.4 | IC50 | 54 | — | |
DVMMSUYWABLYCR
|
7.4 | IC50 | 2 | — | |
GIODDBAYPWNJIQ
|
7.4 | IC50 | 4 | — | |
IYEQRNGTRJYQEW
|
7.4 | Ki | 6 | — | |
JGKOYZSEGMIFTB
|
7.4 | IC50 | 2 | — | |
UQNNJYLAPYGZBD
|
7.4 | Ki | 28 | — | |
BJFMFEYQCRMJSU
|
7.4 | IC50 | 2 | — | |
CPJULNXNBQMSHF
|
7.4 | IC50 | 3 | — | |
GYERFYCOIQWCPP
|
7.4 | Ki | 6 | — | |
ZTPYIOAESPUXFH
|
7.4 | IC50 | 4 | — | |
KRCPKGPVOUOHOW
|
7.4 | IC50 | 3 | — | |
PVGFBLHZPWPMFD
|
7.4 | IC50 | 2 | — | |
XCYATSRJUCZIJR
|
7.4 | IC50 | 7 | Yes | |
BSBQPLUISHJULY
|
7.4 | IC50 | 11 | — | |
HRTYWRWOZZLPDH
|
7.4 | IC50 | 2 | — | |
KRHJQHMWPVTYCU
|
7.4 | IC50 | 6 | — | |
YESKHRZGFKDGEH
|
7.4 | IC50 | 3 | — | |
MJHOMTRKVMKCNE
|
7.3 | IC50 | 12 | — | |
ZDNURMVOKAERHZ
|
7.3 | IC50 | 7 | Yes | |
CJWIBINTCNTMJT
|
7.3 | IC50 | 4 | — | |
COGIYNUARZWUAJ
|
7.3 | IC50 | 2 | — | |
ZXYVWKYLUPYZGL
|
7.3 | Kd | 5 | — | |
ZSHRAUSJZQDIJR
|
7.3 | IC50 | 9 | Yes | |
FTXKUBNATJTYSH
|
7.3 | IC50 | 2 | — | |
FIWNVHIDDOMDBP
|
7.3 | IC50 | 2 | — | |
INTPTKHSGKBHHW
|
7.3 | IC50 | 5 | Yes | |
JOCJOJHKDUXVEF
|
7.3 | IC50 | 2 | — | |
KTUFNOKKBVMGRW
|
7.3 | IC50 | 38 | Yes | |
LVMAULGVWBINFP
|
7.3 | IC50 | 6 | — | |
MLNZPKUVAATQRY
|
7.3 | IC50 | 4 | — | |
PGQWALGGBUYLQF
|
7.3 | IC50 | 12 | — | |
RGNHKJWHFIPHIM
|
7.3 | Ki | 66 | — | |
UDHQGXCXSRGAPA
|
7.3 | IC50 | 4 | — | |
ZCCJKVBTHCOISJ
|
7.3 | Ki | 46 | — |