Target Details
| UniProt AC | P16234 |
|---|---|
| Gene Symbol | PDGFRA |
| Protein Name | Platelet-derived growth factor receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 860
- Clinical molecules 94
- Avg pChEMBL 7.24
KEGG Pathways (22)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Focal adhesion
- Gap junction
- Glioma
- Human cytomegalovirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (4)
Active Molecules (860)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
REDQNEIEGUJUSR
|
7.6 | Ki | 6 | — | |
RQJCPYMTCVHMBN
|
7.6 | Ki | 6 | — | |
HFJIWOVMXXZSKT
|
7.6 | IC50 | 3 | — | |
HTYOBBSZIFVMRH
|
7.6 | Ki | 6 | — | |
JXHVPOHWUDYYJU
|
7.6 | IC50 | 2 | — | |
OQYVAKAMHRACJL
|
7.6 | IC50 | 2 | — | |
ORRHVRJUSPCILV
|
7.6 | Ki | 16 | — | |
PTMRLZVVTLYCDK
|
7.6 | Ki | 6 | — | |
QFOLIEMAGXRGHA
|
7.6 | IC50 | 2 | — | |
SDYGMEWQBSWSIW
|
7.6 | IC50 | 6 | — | |
UECRIUGPTSAZMC
|
7.6 | IC50 | 2 | — | |
WJEOLQLKVOPQFV
|
7.6 | Kd | 24 | — | |
YOHLRCOPRAVUCJ
|
7.6 | IC50 | 6 | — | |
VLCIBPAOYYGWLG
|
7.6 | Ki | 6 | — | |
AOHLFNGYVXMGNP
|
7.6 | Ki | 6 | — | |
BYRBUVTUGSOTSC
|
7.6 | IC50 | 7 | Yes | |
GUBJNPWVIUFSTR
|
7.6 | Kd | 103 | — | |
HRKYCRIVTWSVJU
|
7.6 | IC50 | 4 | Yes | |
JYSCRDCBJSBWKB
|
7.6 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
7.6 | Kd | 153 | — | |
SAEGVASGMTZGFI
|
7.6 | IC50 | 2 | — | |
DPFXYGUGSJIYFI
|
7.6 | Ki | 6 | — | |
FDCKDXZISZRERO
|
7.6 | IC50 | 5 | — | |
KNDPXYAMINMLED
|
7.6 | IC50 | 11 | — | |
VKUNXLBYSBCGAD
|
7.6 | Ki | 6 | — | |
YVVWAUQFCQIDIN
|
7.6 | Ki | 6 | — | |
BRXZUOJFGVQTAB
|
7.5 | IC50 | 3 | Yes | |
FTXKUBNATJTYSH
|
7.5 | IC50 | 2 | — | |
LSJAPABXQBDHRE
|
7.5 | IC50 | 5 | — | |
NGKALCMOLVCFHL
|
7.5 | Kd | 5 | — | |
QXWNDTWKOGDJMG
|
7.5 | IC50 | 5 | — | |
VNBRGSXVFBYQNN
|
7.5 | IC50 | 22 | Yes | |
DCNGPVQCPFIEBU
|
7.5 | IC50 | 2 | — | |
GVQYSEHILFQSHO
|
7.5 | IC50 | 2 | — | |
MIOCXPOZNHTSBC
|
7.5 | IC50 | 2 | — | |
NDEFXZOKPREYOV
|
7.5 | IC50 | 9 | — | |
OOSYGDRIWJDGFV
|
7.5 | IC50 | 2 | — | |
RWZAFECYIQQVPG
|
7.5 | IC50 | 2 | — | |
WOSBNMWHFVPOIW
|
7.5 | IC50 | 2 | — | |
YTHSVVWEPDRWLW
|
7.5 | Ki | 6 | — | |
ZWSUFCVOLVLTHS
|
7.5 | IC50 | 2 | — | |
FWXNEFMIRVAQLN
|
7.5 | IC50 | 4 | — | |
URKLHKCMUZBPEN
|
7.5 | Ki | 6 | — | |
FMCLDFJJIAZKCA
|
7.5 | Kd | 5 | — | |
NEXXSLYFHONHLW
|
7.5 | IC50 | 2 | — | |
NPKCQIBHFHDBIO
|
7.5 | Ki | 6 | — | |
KEDANNMRCOENMZ
|
7.5 | IC50 | 7 | — | |
HBXDLZBPKJEWHZ
|
7.5 | IC50 | 2 | — | |
HFHLYOUFUGWMBG
|
7.5 | Ki | 6 | — | |
NDEFXZOKPREYOV
|
7.5 | IC50 | 8 | — |