Target Details
| UniProt AC | P16234 |
|---|---|
| Gene Symbol | PDGFRA |
| Protein Name | Platelet-derived growth factor receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 860
- Clinical molecules 94
- Avg pChEMBL 7.24
KEGG Pathways (22)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Focal adhesion
- Gap junction
- Glioma
- Human cytomegalovirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (4)
Active Molecules (860)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XESKGZXKYIRKRJ
|
7.8 | Ki | 6 | — | |
MENVZXUPTOFKRC
|
7.8 | IC50 | 3 | — | |
MVPVPEPQINQQJL
|
7.8 | IC50 | 4 | — | |
PLKJJHPCIPKTMV
|
7.8 | IC50 | 2 | — | |
UKYJKXMPIDEQFF
|
7.8 | IC50 | 16 | — | |
AMHUBFWCCMLLCJ
|
7.8 | IC50 | 15 | — | |
DHONEALZRPCJOV
|
7.8 | Ki | 6 | — | |
ZIKJGFZRXYVGMK
|
7.8 | IC50 | 2 | — | |
BWFVHQMKEHJIGA
|
7.7 | Ki | 6 | — | |
FEMXGYPLUJMECJ
|
7.7 | IC50 | 2 | — | |
LYBAWURNJUOHRS
|
7.7 | Ki | 6 | — | |
NVXYJRPMNZXXML
|
7.7 | IC50 | 2 | — | |
OMWAXUAYDHMCSG
|
7.7 | Ki | 6 | — | |
VPWJHKVHKZOWKO
|
7.7 | Ki | 6 | — | |
FHDRORBDPYLAEQ
|
7.7 | Ki | 6 | — | |
QODZCSPDZVDCSD
|
7.7 | IC50 | 7 | — | |
GUUYUIDTJAWAHO
|
7.7 | IC50 | 4 | — | |
IISXSKIQHHGCGE
|
7.7 | Ki | 6 | — | |
BEVNNTNJJJWQAK
|
7.7 | IC50 | 2 | — | |
BQUCMYBIGNGMFC
|
7.7 | IC50 | 5 | — | |
DKFVXLBMKSCYMJ
|
7.7 | Ki | 6 | — | |
DUZZUNRKDFGPSJ
|
7.7 | IC50 | 5 | — | |
GIBYRJLRSLPQGP
|
7.7 | IC50 | 6 | — | |
GZXURVNEOFVVRG
|
7.7 | Ki | 6 | — | |
KXMZDGSRSGHMMK
|
7.7 | IC50 | 14 | — | |
NCCSNHRBEQKRSB
|
7.7 | Ki | 6 | — | |
PAUHYDQXWBOZBD
|
7.7 | IC50 | 4 | — | |
VSVWQTDDGQSGHP
|
7.7 | Ki | 51 | — | |
WDTKJTQWHUMMDU
|
7.7 | IC50 | 2 | — | |
YVRZYHGLKSQXNA
|
7.7 | Ki | 6 | — | |
HGHPBMDBLYJOMZ
|
7.7 | Ki | 6 | — | |
OMVAYCDDPIHBDR
|
7.7 | IC50 | 5 | — | |
DVEKPOFBEAWBKW
|
7.7 | IC50 | 2 | — | |
FRGHNLRLGIIDDA
|
7.7 | IC50 | 2 | — | |
IGVBIRDVFQYICG
|
7.7 | Ki | 6 | — | |
MDFHFYALOAZVKP
|
7.7 | IC50 | 2 | — | |
AISWQGLURAAAKE
|
7.7 | IC50 | 7 | — | |
KVMLMFRXRZLEGU
|
7.6 | IC50 | 4 | — | |
KVTMDRDZMBVWNC
|
7.6 | IC50 | 6 | — | |
ZXAMVJNNDJRGFG
|
7.6 | IC50 | 4 | — | |
BLQYVHBZHAISJM
|
7.6 | IC50 | 21 | Yes | |
CHLFFSKXUJQLQO
|
7.6 | IC50 | 7 | — | |
FIQQIMWSRXTHTA
|
7.6 | IC50 | 2 | — | |
KQCBMFNKIZAQSF
|
7.6 | IC50 | 2 | — | |
LPJDSINAEJVSNX
|
7.6 | IC50 | 6 | Yes | |
OPFGGEANRKOGEG
|
7.6 | Ki | 6 | — | |
RGAHTFBLOZYPNE
|
7.6 | IC50 | 2 | — | |
TXEBERLYUZPASZ
|
7.6 | IC50 | 2 | — | |
AMILNSQCJWLQJG
|
7.6 | IC50 | 3 | — | |
CLWKPYABKROLCK
|
7.6 | Ki | 6 | — |