Target Details
UniProt ACP16234
Gene SymbolPDGFRA
Protein NamePlatelet-derived growth factor receptor alpha
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF07679 (I-set) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr)
Summary
  • Multi-target molecules 860
  • Clinical molecules 94
  • Avg pChEMBL 7.24
Top Co-occurrence Targets
Active Molecules (860)
InChIKey pChEMBL Type Targets Clinical
PKXSPUDURLLHHG 8.1 IC50 5 Yes
ZASMEEJOVACSTK 8.0 Ki 6
CDOQYTRVCWQMJM 8.0 Ki 6
OFTYCXRAQKFFEW 8.0 Ki 6
YYICSPRZBVQPTF 8.0 Ki 6
ZUCUJAOPBDUFMB 8.0 Ki 6
JGWRKYUXBBNENE 8.0 IC50 11
TTYGGHQORNSTIY 8.0 Ki 6
YNFGJAAJMZXYQP 8.0 Ki 6
DYNHJHQFHQTFTP 8.0 IC50 38
HKSZLNNOFSGOKW 8.0 Kd 213
LOLPPWBBNUVNQZ 8.0 IC50 97 Yes
RAHBGWKEPAQNFF 8.0 Kd 26
RWHCDDJSGYJEHN 8.0 IC50 4
SZJRFGYYRZITCZ 8.0 IC50 4
URESLPMFUBHALD 8.0 IC50 2
WUEVFQBRVSPKLA 8.0 IC50 2
XXJWYDDUDKYVKI 8.0 IC50 52
YRUDYNCGPZHXRB 8.0 Kd 6
YVNKPHLJKPWZRT 8.0 IC50 4
KWVDRTIIZKGPOQ 8.0 Ki 6
PIKYCWIZICBHRG 8.0 Ki 6
RCMWTMHAMLWFGA 8.0 Ki 6
WNNZGWZQLJGBNE 8.0 Ki 6
HESUKNSDMPJYHF 8.0 Ki 6
JGEBLDKNWBUGRZ 8.0 IC50 20 Yes
OSKVLQNSYZYKLO 8.0 Ki 6
UKGLXBBBCMZJSW 8.0 Ki 6
ZZGOGKOPTVVJLD 8.0 Ki 6
CFAOCANWUGXOIL 8.0 Ki 6
CVWXJKQAOSCOAB 8.0 Kd 35
WCWUXEGQKLTGDX 8.0 Kd 22 Yes
WDUSDNGPVZEHRQ 8.0 Ki 6
WIXHYLINPBKNTE 8.0 IC50 5 Yes
WJRBHBFXWWGLBI 8.0 Ki 6
ZMYSTIZWTSDYEP 8.0 IC50 5
AVRHXSYMJIZSHR 8.0 Ki 6
KIRQJJFAFLYYJQ 8.0 Ki 6
SSSVBCHLFDKMBI 8.0 Ki 6
WUEKYNCXBMROQI 8.0 Ki 6
UHMOJOLDOBNIHB 7.9 Ki 6
VLIWYQAUGIWSFX 7.9 Ki 6
ABLAJTWOWSSMFU 7.9 IC50 3
FJSAESWYZCNLQU 7.9 Ki 6
HSKISFLIRPOYCF 7.9 IC50 5
KUZBKIYSYFCFOT 7.9 IC50 5
KVBWCMRDDFWCKD 7.9 IC50 2
NGKALCMOLVCFHL 7.9 Kd 5
QCTUWJMAPLGTOR 7.9 IC50 5
QYCFHBDOJSLVRL 7.9 Kd 5
2D structure