Target Details
| UniProt AC | P16234 |
|---|---|
| Gene Symbol | PDGFRA |
| Protein Name | Platelet-derived growth factor receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 860
- Clinical molecules 94
- Avg pChEMBL 7.24
KEGG Pathways (22)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Focal adhesion
- Gap junction
- Glioma
- Human cytomegalovirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (4)
Active Molecules (860)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JGRUAZVMJJCPHI
|
8.2 | IC50 | 2 | — | |
WIVJEMFJDXIPRD
|
8.2 | IC50 | 2 | — | |
CYPOOUITBHWAKE
|
8.2 | IC50 | 4 | — | |
LETIJBVXDGOQFG
|
8.2 | IC50 | 5 | — | |
ODFKDTMBDLHPKM
|
8.2 | IC50 | 2 | — | |
PEPJPELNFRAZNQ
|
8.2 | IC50 | 2 | — | |
UIPHWSFCVAAJDU
|
8.2 | IC50 | 4 | — | |
RITAVMQDGBJQJZ
|
8.2 | Ki | 33 | — | |
NHMWKPIXGXPWGN
|
8.2 | IC50 | 2 | — | |
BLYDOULCQABGHT
|
8.2 | Ki | 6 | — | |
WNMAXXDDBQOLPI
|
8.2 | IC50 | 5 | — | |
HJSPWWLBAHRSAY
|
8.2 | IC50 | 2 | — | |
NYKOXJAXPORIHO
|
8.2 | Ki | 6 | — | |
YTJWRGUFMQLAPJ
|
8.2 | IC50 | 2 | — | |
VHIADSOUXPEWOM
|
8.2 | Ki | 6 | — | |
IFUCZPASJWTYRU
|
8.2 | IC50 | 5 | — | |
IRVGRHMDHCZIOZ
|
8.2 | IC50 | 4 | — | |
JBJZIAHKSVQDAN
|
8.2 | IC50 | 5 | Yes | |
OAFIHAHWHDARSB
|
8.2 | IC50 | 4 | — | |
ROYLPDZGPLFQSV
|
8.2 | IC50 | 3 | — | |
LILXUVCZUBSSFA
|
8.1 | IC50 | 6 | — | |
QMEZKJBCLUGJTN
|
8.1 | IC50 | 5 | — | |
JMVVTEATJVVTPU
|
8.1 | Ki | 6 | — | |
FNVHVYCXTFAQSG
|
8.1 | Ki | 6 | — | |
IONVXRPWTRMITM
|
8.1 | Ki | 6 | — | |
JLFPGEKGHMUMDY
|
8.1 | Ki | 6 | — | |
VTWWRKFUHCSCEW
|
8.1 | Kd | 19 | — | |
XBUZLFQDBPBWCK
|
8.1 | Ki | 6 | — | |
ATWXIAXXSMESBD
|
8.1 | IC50 | 2 | — | |
FTERNYMEXWLTAM
|
8.1 | IC50 | 5 | Yes | |
HKSZLNNOFSGOKW
|
8.1 | Ki | 118 | — | |
MRTHXFZEQBERDI
|
8.1 | IC50 | 11 | — | |
OSZVHJYNXBUVAH
|
8.1 | IC50 | 12 | — | |
PJNSVPCZGALJML
|
8.1 | IC50 | 5 | — | |
PWDPLHOKCYLVIC
|
8.1 | IC50 | 5 | — | |
RTYJMUXLFRYRBU
|
8.1 | Ki | 35 | — | |
UTZFAVQAWTWOKK
|
8.1 | IC50 | 5 | — | |
CPMDPSXJELVGJG
|
8.1 | Ki | 6 | — | |
UDIUFPPEHOBBAN
|
8.1 | Ki | 6 | — | |
XZXHXSATPCNXJR
|
8.1 | IC50 | 165 | Yes | |
HWZNBJUXOVHGSL
|
8.1 | Ki | 6 | — | |
IOXCZKDMVMERGD
|
8.1 | Ki | 6 | — | |
WKQQROGAGZDSBZ
|
8.1 | Ki | 6 | — | |
FGLRXTXAKOMMOX
|
8.1 | IC50 | 5 | — | |
FHTTVJXLZSYAJH
|
8.1 | Ki | 6 | — | |
HXUZQEYFKAZBPX
|
8.1 | IC50 | 4 | Yes | |
JLWGOAGEDWMEBT
|
8.1 | IC50 | 10 | — | |
JLWGOAGEDWMEBT
|
8.1 | IC50 | 10 | — | |
LHKUVOGMYOGQMG
|
8.1 | Ki | 6 | — | |
OPRQSQDMYPVYOV
|
8.1 | IC50 | 7 | — |