Target Details
| UniProt AC | P16234 |
|---|---|
| Gene Symbol | PDGFRA |
| Protein Name | Platelet-derived growth factor receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF25305 (Ig_PDGFR_d4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 860
- Clinical molecules 94
- Avg pChEMBL 7.24
KEGG Pathways (22)
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocytosis
- Focal adhesion
- Gap junction
- Glioma
- Human cytomegalovirus infection
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (4)
Active Molecules (860)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CYVPXDNOIYCAAV
|
8.5 | IC50 | 2 | — | |
DRBIGHXBYOJZLO
|
8.4 | IC50 | 3 | — | |
OMPVQOOIKZDYGO
|
8.4 | IC50 | 2 | — | |
UQLOTEZFDHTNMJ
|
8.4 | IC50 | 2 | — | |
GVFQHBBRWBJGNU
|
8.4 | IC50 | 5 | — | |
SFUSDJRVEVLCSW
|
8.4 | IC50 | 2 | — | |
FEGRQUWSKADGSP
|
8.4 | IC50 | 6 | Yes | |
GFHOQPFRWWTZIG
|
8.4 | IC50 | 2 | — | |
MPVGZUGXCQEXTM
|
8.4 | Kd | 61 | Yes | |
DZFZXPPHBWCXPQ
|
8.4 | IC50 | 12 | — | |
OEUMLQMTMOCCGW
|
8.4 | Kd | 6 | — | |
HMZRSZQIXPNKJY
|
8.4 | IC50 | 4 | — | |
LODWOBAYUQRWKD
|
8.4 | IC50 | 7 | — | |
SEJGTFPOEJWEGG
|
8.3 | Kd | 149 | — | |
AYBLFKIMJMUPEC
|
8.3 | Ki | 6 | — | |
CXQHYVUVSFXTMY
|
8.3 | IC50 | 154 | — | |
LBAQJHGPPPQHFJ
|
8.3 | IC50 | 2 | — | |
INOASWZOZPQAQM
|
8.3 | IC50 | 5 | — | |
CUIHSIWYWATEQL
|
8.3 | Kd | 61 | Yes | |
ACCSYFAQPQXJJO
|
8.3 | Ki | 6 | — | |
ACSSIWPJCYCXGD
|
8.3 | IC50 | 4 | — | |
IQCIFDSCWKQXJA
|
8.3 | IC50 | 4 | — | |
JAXRQZOMEYHMHJ
|
8.3 | IC50 | 2 | — | |
KSELTIXXASIVDL
|
8.3 | IC50 | 2 | — | |
KVDZJYLUBBYJIX
|
8.3 | IC50 | 2 | — | |
NQVBNOPSVRCGSI
|
8.3 | IC50 | 2 | — | |
YIQKRGSTCNRKES
|
8.3 | Ki | 6 | — | |
YXZQRTLGEGYVTJ
|
8.3 | IC50 | 2 | — | |
NCPIMEOPSFOWKB
|
8.3 | IC50 | 4 | — | |
XPBJIFLFRWUBPO
|
8.3 | IC50 | 3 | — | |
AQAZMVVLAOLUPL
|
8.3 | IC50 | 2 | — | |
BHJMKBAJRGNMGC
|
8.3 | IC50 | 2 | — | |
CDDZQGUAUSHZFZ
|
8.3 | IC50 | 2 | — | |
FKNPENIHAAPMRC
|
8.3 | IC50 | 2 | — | |
GMUXDKZNMOZDKO
|
8.3 | IC50 | 2 | — | |
HTIOELJVBGXYQR
|
8.3 | IC50 | 2 | — | |
IQQVFGJWEJAHBR
|
8.3 | IC50 | 2 | — | |
KLOPQHWNVNJIMS
|
8.3 | IC50 | 2 | — | |
LQEFORQTPQKHOT
|
8.3 | IC50 | 2 | — | |
MKFKYKXIANOUHV
|
8.3 | IC50 | 2 | — | |
MPDVLCDGYNYLDZ
|
8.3 | IC50 | 2 | — | |
TXNMFHSHEJRKSX
|
8.3 | IC50 | 2 | — | |
XBCQOKINRQAZKD
|
8.3 | IC50 | 2 | — | |
YVRJNNUMUYEWAJ
|
8.3 | IC50 | 2 | — | |
YWSJCLQQBSHJBQ
|
8.3 | IC50 | 2 | — | |
YZRLWPBYTMKRQR
|
8.3 | IC50 | 11 | — | |
ZGLBORDNOBELSS
|
8.3 | IC50 | 2 | — | |
MPYUMMWCLQVMLG
|
8.2 | IC50 | 11 | — | |
VAARYSWULJUGST
|
8.2 | Kd | 119 | Yes | |
BVSYMJUCSKOBAS
|
8.2 | IC50 | 2 | — |