Target Details
| UniProt AC | P16066 |
|---|---|
| Gene Symbol | NPR1 |
| Protein Name | Atrial natriuretic peptide receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01094 (ANF_receptor) PF00211 (Guanylate_cyc) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 19
- Clinical molecules 0
- Avg pChEMBL 8.15
KEGG Pathways (11)
Active Molecules (19)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QGFSVPWZEPKNDV
|
10.3 | IC50 | 3 | — | |
DKENAONXZOBIFG
|
10.0 | IC50 | 2 | — | |
MVVBMTAWECNSCX
|
10.0 | Ki | 2 | — | |
AYCBRUDZNRVKGK
|
9.6 | Ki | 3 | — | |
AYCBRUDZNRVKGK
|
9.5 | IC50 | 3 | — | |
VKNFJABNSMOWGE
|
9.5 | Ki | 2 | — | |
FUVHGJXBAITLDM
|
9.4 | Ki | 2 | — | |
SMLLMWDCKCAQKV
|
9.3 | Ki | 2 | — | |
NSQLIUXCMFBZME
|
9.2 | Ki | 2 | — | |
UXLDAJPPNWDHHB
|
7.4 | IC50 | 3 | — | |
CGIAJIVLXUYRPS
|
7.3 | IC50 | 3 | — | |
LLIWCAYHKZUTHH
|
7.2 | Ki | 2 | — | |
USKHZVUKGMGKMN
|
7.2 | Ki | 2 | — | |
BFCFDUDISIBVNN
|
7.1 | Ki | 2 | — | |
WTSQMOAJTSQRKS
|
6.9 | IC50 | 2 | — | |
MCHMSEFZIGFZBO
|
6.4 | Ki | 2 | — | |
WNMJJSOJFSGNGI
|
6.3 | Ki | 2 | — | |
UWAQSJWJCXAOOI
|
6.2 | Ki | 2 | — | |
BNWIVWQCCFRSQN
|
6.1 | IC50 | 16 | — |