Target Details
| UniProt AC | P15917 |
|---|---|
| Gene Symbol | lef |
| Protein Name | Lethal factor |
| Organism | Bacillus anthracis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF09156 (Anthrax-tox_M) PF07737 (ATLF) |
Summary
- Multi-target molecules 16
- Clinical molecules 2
- Avg pChEMBL 7.74
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PVPXSRWESCVIBD
|
9.9 | Ki | 2 | — | |
QKBHUOCFQAXIBG
|
9.8 | Ki | 3 | — | |
BPGDVHWVHMDFBK
|
9.6 | Ki | 2 | — | |
RKZDOJQKLCPUQZ
|
9.5 | Ki | 2 | — | |
AWFIZJRPXRHSEA
|
9.0 | Ki | 2 | — | |
DUBRLRRJAJGWMU
|
8.9 | Ki | 3 | — | |
LUCFRFDOOYLALP
|
7.3 | IC50 | 4 | Yes | |
SWPCXTNDGTURLE
|
7.2 | Ki | 3 | — | |
INIOOWZLISZDKY
|
7.0 | IC50 | 2 | — | |
KICRIIPFHBTWCQ
|
6.9 | IC50 | 2 | — | |
UOLICGDBHYFWJG
|
6.7 | IC50 | 2 | — | |
NLTKRFJIWZFZTF
|
6.7 | IC50 | 2 | — | |
JMCIPOCGNQTZQT
|
6.6 | IC50 | 2 | — | |
ILGJGLKILKMTFU
|
6.4 | IC50 | 2 | — | |
PGBHMTALBVVCIT
|
6.3 | Ki | 59 | — | |
SUEBJDNLBVTIQP
|
6.0 | IC50 | 8 | Yes |