Target Details
| UniProt AC | P15735 |
|---|---|
| Gene Symbol | PHKG2 |
| Protein Name | Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 76
- Clinical molecules 11
- Avg pChEMBL 6.69
KEGG Pathways (3)
Associated Diseases (3)
Active Molecules (76)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.8 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
9.3 | IC50 | 408 | — | |
KOZFSFOOLUUIGY
|
8.8 | IC50 | 88 | Yes | |
UIARLYUEJFELEN
|
8.8 | Kd | 289 | Yes | |
WINHZLLDWRZWRT
|
8.2 | Kd | 201 | Yes | |
FZBVNCFBCNXULH
|
8.2 | IC50 | 18 | — | |
BSFNGHCTZDCQBF
|
7.9 | Ki | 93 | — | |
QQWUGDVOUVUTOY
|
7.9 | Kd | 231 | Yes | |
WINHZLLDWRZWRT
|
7.8 | Ki | 66 | — | |
MWKSRKSEWLRPBL
|
7.8 | Kd | 1075 | — | |
OWRXHGAFWZFFCW
|
7.3 | Ki | 113 | — | |
AYCPARAPKDAOEN
|
7.3 | Kd | 73 | — | |
NXSJMRCTGYTSTK
|
7.2 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
7.1 | Kd | 170 | — | |
MVJMMLFMPWITEJ
|
7.1 | Ki | 110 | — | |
ADMFLILDQJSEIK
|
7.0 | Ki | 72 | — | |
CTNPALGJUAXMMC
|
7.0 | Kd | 151 | — | |
AILRADAXUVEEIR
|
7.0 | IC50 | 75 | — | |
LRZYYIZFBXFSJB
|
6.9 | Ki | 69 | — | |
ZCCPLJOKGAACRT
|
6.9 | Kd | 599 | — | |
YYLKKYCXAOBSRM
|
6.8 | Kd | 191 | — | |
GCYXEGSPUDSZJY
|
6.8 | Ki | 82 | — | |
RJZDECGDCKOHBV
|
6.8 | Ki | 70 | — | |
XPHWIERLJBFPFV
|
6.8 | Ki | 69 | — | |
FUMCKNCUEAQHCV
|
6.7 | Ki | 103 | — | |
PCQMERRARZKTPW
|
6.7 | Ki | 68 | — | |
MJHOMTRKVMKCNE
|
6.7 | IC50 | 12 | — | |
DBXGGXLBTWZXBB
|
6.6 | Ki | 39 | — | |
JZTOUVBEZONDKA
|
6.6 | Ki | 80 | — | |
OADRBDVURCEKRP
|
6.6 | Ki | 44 | — | |
RYYNGWLOYLRZLK
|
6.6 | Ki | 104 | — | |
UDFDIIVNIYWXDM
|
6.6 | Ki | 74 | — | |
VBIYDORVDCFKHM
|
6.6 | Ki | 13 | — | |
XZXHXSATPCNXJR
|
6.6 | Kd | 165 | Yes | |
AWDORCFLUJZUQS
|
6.5 | Ki | 22 | — | |
PNKALLUVKOKYHZ
|
6.5 | Ki | 32 | — | |
SQXSMLLCDWJNAC
|
6.5 | Ki | 20 | — | |
UYJNQQDJUOUFQJ
|
6.5 | Ki | 68 | — | |
ZGZVRPRSFXRGCF
|
6.5 | Ki | 76 | — | |
HHZIURLSWUIHRB
|
6.5 | Kd | 57 | Yes | |
DKZYXHCYPUVGAF
|
6.4 | Kd | 112 | — | |
LRINYHMQZRENCY
|
6.4 | Ki | 29 | — | |
OLVBAUVSICCWEJ
|
6.4 | Ki | 39 | — | |
QYGMZFLXMWJYRJ
|
6.4 | Ki | 14 | — | |
ZWVZORIKUNOTCS
|
6.4 | Ki | 69 | — | |
OUSFTKFNBAZUKL
|
6.3 | Kd | 58 | Yes | |
ULXXDDBFHOBEHA
|
6.3 | Kd | 15 | Yes | |
KRIUNPBAQZGFQA
|
6.3 | Kd | 76 | — | |
GLMWKEAUVZDGKE
|
6.3 | Ki | 23 | — | |
CMWRPDHVGMHLSZ
|
6.3 | IC50 | 22 | — |