Target Details
| UniProt AC | P15328 |
|---|---|
| Gene Symbol | FOLR1 |
| Protein Name | Folate receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03024 (Folate_rec) |
Summary
- Multi-target molecules 56
- Clinical molecules 2
- Avg pChEMBL 8.57
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (56)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HHKAOUMVRGSKLS
|
12.3 | Kd | 2 | — | |
KXVFDIDJQOTBSL
|
11.7 | Kd | 2 | — | |
HHKAOUMVRGSKLS
|
11.5 | Kd | 2 | — | |
WMTFSFGBNBUALY
|
9.8 | IC50 | 5 | — | |
NQIQMFMYULMMGE
|
9.8 | Kd | 2 | — | |
UNSSSMUKJOLMJV
|
9.5 | IC50 | 5 | — | |
VCNJYHGDMDELAI
|
9.5 | IC50 | 2 | — | |
WMBYSCVMFMNUQV
|
9.5 | IC50 | 5 | — | |
JWZBILLJZHUAOY
|
9.4 | IC50 | 5 | — | |
QSMJJFQXDNSFGZ
|
9.4 | Kd | 2 | — | |
QXWUFUZJYLBZQF
|
9.4 | IC50 | 3 | — | |
HPAURQDCTYKMTE
|
9.3 | IC50 | 4 | — | |
BDXBDXZHMOFNOY
|
9.2 | IC50 | 3 | — | |
ZGMCQEIDLHETAQ
|
9.2 | Kd | 2 | — | |
JXLUUFBZGXCZRH
|
9.2 | Kd | 2 | — | |
STQPVYHCDNSBIJ
|
9.2 | IC50 | 5 | — | |
UEVAKXKCGSGJIG
|
9.0 | IC50 | 2 | — | |
JXLUUFBZGXCZRH
|
9.0 | Kd | 2 | — | |
FTSMBZFBGMYYIT
|
9.0 | IC50 | 5 | — | |
SIDIEQMDPONVCD
|
9.0 | IC50 | 3 | — | |
VEKHZPVGFDPVJG
|
9.0 | IC50 | 5 | — | |
FSOJIOKMUXQEMI
|
8.9 | IC50 | 5 | — | |
RNDCKROBKFEYEB
|
8.8 | IC50 | 2 | — | |
STXAYXIUQRNEBG
|
8.8 | IC50 | 3 | — | |
WGEYLZWUJAEXSI
|
8.8 | IC50 | 2 | — | |
PNRJTEIZPOHDEE
|
8.8 | IC50 | 2 | — | |
ADFLVKAWSSGDBU
|
8.7 | IC50 | 3 | — | |
VFYUKZOGWIMWFW
|
8.7 | IC50 | 5 | — | |
VMGGIKVXYOZFJO
|
8.6 | IC50 | 4 | — | |
IFTGJDSAOAUHRL
|
8.6 | IC50 | 2 | — | |
CYOOKDIMCAPJGV
|
8.5 | IC50 | 5 | — | |
UFNWIIALSMNORN
|
8.5 | IC50 | 5 | — | |
QLSVPQAGJDLITE
|
8.4 | IC50 | 5 | — | |
VKYMIASYZYDIRX
|
8.4 | IC50 | 2 | — | |
UPENPAQNDNZZTP
|
8.3 | IC50 | 5 | — | |
QNFVXICXLFWABV
|
8.2 | IC50 | 3 | — | |
CEPQCJFDTGQKDN
|
8.2 | IC50 | 4 | — | |
VLHCBXFJXATDOK
|
8.2 | IC50 | 2 | — | |
SNKVTLINZXZOGT
|
8.2 | IC50 | 2 | — | |
KVBZUTNKUVNMNN
|
8.1 | IC50 | 3 | — | |
NDBHIBYSTUVPRS
|
8.0 | IC50 | 3 | — | |
LYDGQYDYRQVOBF
|
8.0 | IC50 | 2 | — | |
IVTVGDXNLFLDRM
|
7.8 | IC50 | 8 | — | |
OUMBMSSXXWAJDS
|
7.8 | IC50 | 3 | — | |
RMEHPWHLFJJYTB
|
7.8 | IC50 | 5 | — | |
WBXPDJSOTKVWSJ
|
7.4 | IC50 | 10 | Yes | |
ARIQPXNXGFKWNW
|
7.3 | IC50 | 3 | — | |
JLRJTWXBYRMGEB
|
7.3 | IC50 | 4 | — | |
HQPQAUMWVMDRCN
|
7.0 | IC50 | 3 | — | |
RPXDQPDLDPKBHG
|
6.9 | Kd | 3 | Yes |