Target Details
| UniProt AC | P15153 |
|---|---|
| Gene Symbol | RAC2 |
| Protein Name | Ras-related C3 botulinum toxin substrate 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00071 (Ras) |
Summary
- Multi-target molecules 3
- Clinical molecules 0
- Avg pChEMBL 7.14
KEGG Pathways (31)
- Adherens junction
- Axon guidance
- B cell receptor signaling pathway
- Cadherin signaling
- Chemokine signaling pathway
- Choline metabolism in cancer
- Colorectal cancer
- Diabetic cardiomyopathy
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Integrin signaling
- Leukocyte transendothelial migration
- MAPK signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Pancreatic cancer
- Pathways in cancer
- Prion disease
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Sphingolipid signaling pathway
- VEGF signaling pathway
- Viral myocarditis
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (3)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MIDUFIRTIFUTQA
|
7.2 | Kd | 3 | — | |
MWKSRKSEWLRPBL
|
7.2 | Kd | 1075 | — | |
LJCANTASZGYJLG
|
7.0 | IC50 | 4 | — |