Target Details
| UniProt AC | P15056 |
|---|---|
| Gene Symbol | BRAF |
| Protein Name | Serine/threonine-protein kinase B-raf |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF07714 (PK_Tyr_Ser-Thr) PF02196 (RBD) |
Summary
- Multi-target molecules 2,643
- Clinical molecules 78
- Avg pChEMBL 7.81
KEGG Pathways (44)
- Acute myeloid leukemia
- Alcoholism
- Alzheimer disease
- Bladder cancer
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Chronic myeloid leukemia
- Colorectal cancer
- Cushing syndrome
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gastric cancer
- Glioma
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Insulin signaling pathway
- Long-term depression
- Long-term potentiation
- MAPK signaling pathway
- Melanoma
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Renal cell carcinoma
- Serotonergic synapse
- Thyroid cancer
- Vascular smooth muscle contraction
- cAMP signaling pathway
- mTOR signaling pathway
Associated Diseases (10)
Active Molecules (2,643)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GWWMADPPWXLUER
|
8.8 | IC50 | 2 | — | |
ROTJLNFGZWQSGH
|
8.8 | IC50 | 2 | — | |
SWYMZYAYCOOLSG
|
8.8 | IC50 | 2 | — | |
TYGWPUNSOFXZIP
|
8.8 | IC50 | 2 | — | |
UFJILEUJRRXOHJ
|
8.8 | IC50 | 2 | — | |
WQXODHHFTYPTME
|
8.8 | IC50 | 5 | — | |
YBQICLDGWWEPMS
|
8.8 | IC50 | 2 | — | |
YHJYMZWMIXBQNX
|
8.8 | IC50 | 2 | — | |
YULMIWVPBRHYSJ
|
8.8 | IC50 | 2 | — | |
YWXHCAQISAEKBP
|
8.8 | IC50 | 2 | — | |
ZBUVKZFJRCJJKF
|
8.8 | IC50 | 3 | — | |
LHQUZYBPZRBVPU
|
8.8 | IC50 | 2 | — | |
RSDYZQKJYMWKCT
|
8.8 | IC50 | 2 | — | |
GUWXGAXEMXDUDP
|
8.8 | IC50 | 2 | — | |
ATMWTCHMTMDCOQ
|
8.7 | IC50 | 2 | — | |
BGCVKYSWJAYBBI
|
8.7 | IC50 | 2 | — | |
BRIAZOQJCABKIH
|
8.7 | IC50 | 2 | — | |
BSMCAPRUBJMWDF
|
8.7 | IC50 | 4 | — | |
DVBQSUVLJKVUBQ
|
8.7 | IC50 | 2 | — | |
FOLVBVJHOLIIRE
|
8.7 | IC50 | 2 | — | |
GQKRUHLMMBPTEC
|
8.7 | IC50 | 2 | — | |
GRNQCTMTIYRPGV
|
8.7 | IC50 | 2 | — | |
HJEAPQLJRHRRQR
|
8.7 | IC50 | 2 | — | |
IURUCQHKNQXJDY
|
8.7 | IC50 | 2 | — | |
JNUVEXMQPTVVSO
|
8.7 | IC50 | 2 | — | |
KAXVMMMCHWWRKM
|
8.7 | IC50 | 2 | — | |
KOHWMDVRLFFKNM
|
8.7 | IC50 | 2 | — | |
KUWINQJYGACLDX
|
8.7 | IC50 | 2 | — | |
LEKITHGJJJVYSN
|
8.7 | IC50 | 2 | — | |
OREGPRREBGYGBQ
|
8.7 | IC50 | 2 | — | |
QBSGBBKYIBHYLQ
|
8.7 | IC50 | 2 | — | |
SZSHXYPGPBQNKS
|
8.7 | IC50 | 2 | — | |
VCRWYFQGTCFZDJ
|
8.7 | IC50 | 2 | — | |
XNMKLOSTCLYASB
|
8.7 | IC50 | 2 | — | |
AUMCDHXOXBVWPP
|
8.7 | IC50 | 2 | — | |
FFJPMZAIZAHGTD
|
8.7 | IC50 | 2 | — | |
HCXYJDIXGYPPPH
|
8.7 | IC50 | 2 | — | |
HKLXIGLBNKMGOD
|
8.7 | IC50 | 2 | — | |
JDBHGMBVFCNSHY
|
8.7 | IC50 | 2 | — | |
LDTUEQNAYCVAAO
|
8.7 | IC50 | 2 | — | |
LZGGFVXWAVXQLA
|
8.7 | IC50 | 2 | — | |
PTEZLRAAYJQGKF
|
8.7 | IC50 | 2 | — | |
UDUXYHUWFANFEJ
|
8.7 | IC50 | 2 | — | |
ZMPLUUUXFORXDW
|
8.7 | IC50 | 2 | — | |
CPQCRZXCFJSDSG
|
8.7 | IC50 | 2 | — | |
DNRCPBXFJDGSBQ
|
8.7 | IC50 | 2 | — | |
GAIGZMYWYVKPKA
|
8.7 | IC50 | 2 | — | |
GAQBWXSEJOHZJS
|
8.7 | IC50 | 2 | — | |
GGGFTTMBYHTHTO
|
8.7 | IC50 | 2 | — | |
GJBWANRWQWONGM
|
8.7 | IC50 | 2 | — |