Target Details
| UniProt AC | P15056 |
|---|---|
| Gene Symbol | BRAF |
| Protein Name | Serine/threonine-protein kinase B-raf |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF07714 (PK_Tyr_Ser-Thr) PF02196 (RBD) |
Summary
- Multi-target molecules 2,643
- Clinical molecules 78
- Avg pChEMBL 7.81
KEGG Pathways (44)
- Acute myeloid leukemia
- Alcoholism
- Alzheimer disease
- Bladder cancer
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Chronic myeloid leukemia
- Colorectal cancer
- Cushing syndrome
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gastric cancer
- Glioma
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Insulin signaling pathway
- Long-term depression
- Long-term potentiation
- MAPK signaling pathway
- Melanoma
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Renal cell carcinoma
- Serotonergic synapse
- Thyroid cancer
- Vascular smooth muscle contraction
- cAMP signaling pathway
- mTOR signaling pathway
Associated Diseases (10)
Active Molecules (2,643)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UEFAPHOCMPHIDW
|
9.2 | IC50 | 2 | — | |
WQXYUSBTQMBASI
|
9.2 | IC50 | 2 | — | |
WZILZCPNZNQCRS
|
9.2 | IC50 | 2 | — | |
XCURDAWHBBABCE
|
9.2 | IC50 | 2 | — | |
YJAAENGSEJKFCT
|
9.2 | IC50 | 2 | — | |
PYCRDHRFOVBBQM
|
9.2 | IC50 | 2 | — | |
XMKZIAJYFCXPPO
|
9.2 | IC50 | 2 | — | |
AQZNVPIHZFYWPU
|
9.2 | IC50 | 2 | — | |
OYRCPJFWDDYQRG
|
9.2 | IC50 | 2 | — | |
QJYIMGVDSRUSLN
|
9.2 | IC50 | 2 | — | |
UFRNWXTUQZQHEB
|
9.2 | IC50 | 2 | — | |
ZPMMEQLJGQJSKJ
|
9.2 | IC50 | 2 | — | |
NBTHXUSRXBOARD
|
9.2 | IC50 | 2 | — | |
IBINNYRGHRQIFO
|
9.2 | IC50 | 2 | — | |
NRUJDQAGOKDQBH
|
9.2 | IC50 | 3 | — | |
BTXSFXPMDZDEKQ
|
9.2 | IC50 | 2 | — | |
CLJJOJZHQFORCB
|
9.2 | IC50 | 3 | — | |
KCRBKRJYKPPDNG
|
9.2 | IC50 | 2 | — | |
KEMDLZNSHOZIMO
|
9.2 | IC50 | 2 | — | |
KPBPKIMSIANJOA
|
9.2 | IC50 | 2 | — | |
LDWLKZFOTRFNQS
|
9.2 | IC50 | 2 | — | |
NKVPTHCZFKPFLR
|
9.2 | IC50 | 2 | — | |
NSQSHHMJVMLITG
|
9.2 | IC50 | 2 | — | |
OIYIRZYUSQJZTH
|
9.2 | IC50 | 2 | — | |
PELRAOUKKKUGBN
|
9.2 | IC50 | 2 | — | |
SHWXNUIJYINNCK
|
9.2 | IC50 | 2 | — | |
XASCATHLORIIEH
|
9.2 | IC50 | 2 | — | |
ZWLYLYAHGLYJPE
|
9.2 | IC50 | 2 | — | |
KQBACBRUHFGIHB
|
9.1 | IC50 | 2 | — | |
GZEIUQBPVOBYNA
|
9.1 | IC50 | 2 | — | |
BZHGOIYVJUGAQI
|
9.1 | IC50 | 3 | — | |
GLQHXZGNENSPJX
|
9.1 | IC50 | 2 | — | |
NVLNBEBFJGSCJK
|
9.1 | IC50 | 2 | — | |
FMAPRDUFFLBURT
|
9.1 | IC50 | 2 | — | |
HQSBUBYPWIUFIL
|
9.1 | IC50 | 2 | — | |
XQNRCPXMLMNNPS
|
9.1 | IC50 | 2 | — | |
YFGBLRZGYKYFOK
|
9.1 | IC50 | 2 | — | |
BSPOTOGQWINOGT
|
9.1 | IC50 | 2 | — | |
BYOVYFARSYCHOS
|
9.1 | IC50 | 2 | — | |
DMOUEXIMXNPRQR
|
9.1 | IC50 | 2 | — | |
DZYQLRIKVLHQEF
|
9.1 | IC50 | 2 | — | |
GJPGNFNVUJLBQZ
|
9.1 | IC50 | 2 | — | |
GXCZMYTUQJAGAX
|
9.1 | IC50 | 2 | — | |
IBQHTAUNXNWAJI
|
9.1 | IC50 | 2 | — | |
JODNXTZRZICRLH
|
9.1 | IC50 | 2 | — | |
JOIYVAOMEJSCBK
|
9.1 | IC50 | 2 | — | |
KHSZTGIXNYRJRU
|
9.1 | IC50 | 2 | — | |
NSQMFMWJEYFCCI
|
9.1 | IC50 | 2 | — | |
OCCGPFVCKGXCHU
|
9.1 | IC50 | 2 | — | |
OZOPEVNRONREIV
|
9.1 | IC50 | 2 | — |