Target Details
| UniProt AC | P15056 |
|---|---|
| Gene Symbol | BRAF |
| Protein Name | Serine/threonine-protein kinase B-raf |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF07714 (PK_Tyr_Ser-Thr) PF02196 (RBD) |
Summary
- Multi-target molecules 2,643
- Clinical molecules 78
- Avg pChEMBL 7.81
KEGG Pathways (44)
- Acute myeloid leukemia
- Alcoholism
- Alzheimer disease
- Bladder cancer
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Chronic myeloid leukemia
- Colorectal cancer
- Cushing syndrome
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gastric cancer
- Glioma
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Insulin signaling pathway
- Long-term depression
- Long-term potentiation
- MAPK signaling pathway
- Melanoma
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Renal cell carcinoma
- Serotonergic synapse
- Thyroid cancer
- Vascular smooth muscle contraction
- cAMP signaling pathway
- mTOR signaling pathway
Associated Diseases (10)
Active Molecules (2,643)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IQARZQCIIDWYSQ
|
8.7 | IC50 | 2 | — | |
KZCBXFJPHWUWFQ
|
8.7 | IC50 | 2 | — | |
SBHUAUMYQMOGOC
|
8.7 | IC50 | 2 | — | |
UIDLNSPVAIBRJS
|
8.7 | IC50 | 2 | — | |
VUBFULNSSXNSJT
|
8.7 | IC50 | 2 | — | |
WUHCLCRCBCBJQT
|
8.7 | IC50 | 2 | — | |
YBVLKMMGWXPQRX
|
8.7 | IC50 | 2 | — | |
AHXHPSNGFWTQPX
|
8.7 | IC50 | 2 | — | |
AIPRPSWGJJAMMI
|
8.7 | IC50 | 2 | — | |
NMGUFZZZFPOLHX
|
8.7 | IC50 | 2 | — | |
NTQDRNKJUSQTEG
|
8.7 | IC50 | 2 | — | |
YQWYOOFOVOSYHX
|
8.7 | IC50 | 2 | — | |
ZPFKPMWFOSWJLV
|
8.7 | IC50 | 2 | — | |
AQHIGRWVPFAESP
|
8.7 | IC50 | 2 | — | |
BALNMMOLSVQPFQ
|
8.7 | IC50 | 2 | — | |
BARRZGQMKZYTJV
|
8.7 | IC50 | 2 | — | |
DCTIKIWYRXDSOC
|
8.7 | pIC50 | 2 | Yes | |
DFIVZWWMRMZVLA
|
8.7 | IC50 | 2 | — | |
FRLQZRDDFJVTJS
|
8.7 | IC50 | 3 | — | |
GCVLGXWDFGPGDP
|
8.7 | IC50 | 2 | — | |
HKDMNDSYJYCJAJ
|
8.7 | IC50 | 2 | — | |
HXALSNAYPNDDSO
|
8.7 | IC50 | 3 | — | |
IIFWSFBWNGNUAF
|
8.7 | IC50 | 2 | — | |
IQNUESPLCMDNRV
|
8.7 | IC50 | 3 | — | |
IRCLZLJAEFQVQA
|
8.7 | IC50 | 2 | — | |
IVLPNLXFDCHLKA
|
8.7 | IC50 | 3 | — | |
IWIONOUUGJGBPE
|
8.7 | IC50 | 2 | — | |
JNEGWVZMAAXSDR
|
8.7 | IC50 | 2 | — | |
KKCJMVOTVSOBJV
|
8.7 | IC50 | 3 | — | |
KKVYYGGCHJGEFJ
|
8.7 | IC50 | 6 | Yes | |
KYDSKCOSDPLKLI
|
8.7 | IC50 | 2 | — | |
LGZWNNOKMRSOFV
|
8.7 | IC50 | 2 | — | |
LOPFFGYJBIMBSE
|
8.7 | IC50 | 3 | — | |
MAEIMZUQBHFKFG
|
8.7 | IC50 | 3 | — | |
MFJJLZIXKPDJHY
|
8.7 | IC50 | 2 | — | |
MRONWWYUJGYEFK
|
8.7 | IC50 | 3 | — | |
NKPAXDYLOKPXNV
|
8.7 | IC50 | 2 | — | |
OGFOENLUWIJPAQ
|
8.7 | IC50 | 3 | — | |
OQADNYQXVWLBPF
|
8.7 | IC50 | 3 | — | |
OQPWKRIFJWBPSI
|
8.7 | IC50 | 3 | — | |
PCTIECVOHLCQSU
|
8.7 | IC50 | 3 | — | |
PFBMPRTYJZBTQO
|
8.7 | IC50 | 2 | — | |
PSHYIXJXMAODDE
|
8.7 | IC50 | 2 | — | |
RSMGUCWXMLOUPS
|
8.7 | IC50 | 2 | — | |
SGZHLFXKVNMWRZ
|
8.7 | IC50 | 3 | — | |
UPUBHFBOYYXILS
|
8.7 | IC50 | 3 | — | |
WKHLVCIENFFXAL
|
8.7 | IC50 | 2 | — | |
WUNPJNPKZVFAEX
|
8.7 | IC50 | 2 | — | |
XLZSBGWFJTXBDS
|
8.7 | IC50 | 2 | — | |
ZFEIDQHEBUDXPF
|
8.7 | IC50 | 2 | — |