Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
YRHWMEGQCCRQAT 8.1 Ki 2
ZHLQLUZELIBEJT 8.1 Ki 2
GIWWJSXACMYFKV 8.1 Ki 2
JANXKKALWNYMDP 8.1 Ki 3
MZBKUGGHNJCZTE 8.1 Ki 2
XGJLRKVQXMSBJW 8.1 IC50 16
DEOUAHSUIKDCLJ 8.0 Ki 2
UBZQMNGVBPUKCE 8.0 Ki 4
UNJFTNACNPGPEC 8.0 Ki 6
FLEQTIDRWGGTRR 8.0 Ki 7
GMPMVFUXLJTJET 8.0 Ki 2
HMQQCASSOWMONY 8.0 Ki 2
NBHUXHWJYCGLNS 8.0 Ki 2
STIAETBDCMTLLC 8.0 Ki 2
KWPOKTUWXDCATM 8.0 IC50 16
TVKPVFXZZBBIAN 8.0 Ki 2
YKKWBLSUYZOORV 8.0 Ki 6
YVPJMZCJVHJOFG 8.0 Ki 7
HQJSGBKPXYZTRN 8.0 IC50 16
IKZRLIUEIZSYGZ 8.0 Ki 2
INJYZJLFMOYBRK 8.0 Ki 2
MBZNSAJBODIJCK 8.0 IC50 16
MZTRNWROWIGTRB 8.0 Ki 7
PFAUXAQOEJBLRX 8.0 Ki 4
PSDFROGPPFTBND 8.0 Ki 7
SIPHVHFVEKBHKT 8.0 Ki 7
TURQHSQKHGLRSX 8.0 Ki 2
UGHWRPXZRCYTTI 8.0 Ki 6
VQAWSSJLGHVFHE 8.0 Ki 6
XDEHJKJHEDWFEK 8.0 Ki 2
VDLZNMPWETXSHJ 8.0 Ki 2
HHTMTQUAFKAYSU 8.0 Ki 2
HOMGIOZFYSJYAP 8.0 Ki 2
IZIWQEMYKBYTJE 8.0 Ki 2
KRBLTADBSGBJIF 8.0 Ki 2
OUAMKNYCLUPDQV 8.0 Ki 2
CIGLLASOKXAMLS 8.0 Ki 7
DKSWXNFPYZCJFU 8.0 Ki 6
HFPZDEHIDKJZSN 8.0 Ki 16
LGRQUGHDTPHNOB 8.0 Ki 6
LMJMBPXKXWIKQK 8.0 IC50 16
MFZNONRIQYSLMZ 8.0 Ki 6
NNHRCSJWUBQYQV 8.0 IC50 16
PKJGSRHYDOGGLB 8.0 Ki 17
PTJXEJYDOYCHOL 8.0 IC50 3
UBZGCHSBAOJHLE 8.0 Ki 3
DPSSGGDIOTWPAP 8.0 Ki 2
IXGIOXIKQZCZIK 8.0 Ki 8
JLMKWODKTUEGMY 8.0 Ki 2
LZAOMRNXXVBOBL 8.0 Ki 2
2D structure