Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
TWQAQMSDCDNDFY 8.2 Ki 2
VPZOLJKOURRVNO 8.2 IC50 3
WMCJJXHYPNOCMT 8.2 IC50 16
YIPXEQDLFGBASS 8.2 Ki 5
ZRPUPUBWCXFOCY 8.2 Ki 16
BGRWSFIQQPVEML 8.1 Ki 6
JAUWZXFLIUKTGH 8.1 Ki 4
JFQBVKGJWWZLHU 8.1 Ki 2
OJYWDSGHQXTNRR 8.1 Ki 2
OWTXLWRGHNAFHX 8.1 Ki 6
QMARBOVOPHNZOR 8.1 Ki 2
UKGVLKDJTMUFNB 8.1 Ki 6
UMNMVUGGTKAKKC 8.1 Ki 5
VUSVWZBQTTWZGJ 8.1 Ki 5
WPSKGYBCTJQZGB 8.1 Ki 2
QQIVOICVQUEJEG 8.1 Ki 4
DWEPHBCGVLXMBR 8.1 Ki 5
FUXYUWJJJCFFSW 8.1 Ki 2
GADIKQPUNWAMEB 8.1 Ki 5
LMTLCLNZGQDMAJ 8.1 Ki 2
SWLOMELGJKUNSM 8.1 Ki 2
YUBXINUNAGILPI 8.1 Ki 2
HJYLTAKIKUDBOO 8.1 Ki 2
HRNSOLSYHZMSCD 8.1 Ki 6
KJPFVEHEGGIJIJ 8.1 Ki 4
ORZSFKNQZNYIGS 8.1 Ki 2
DKCAUMRZSZVJCP 8.1 Ki 16
FHVJNRCGUUPETA 8.1 Ki 2
GIATTYVTHLBQCS 8.1 Ki 2
IVGTVZGLPHBTJV 8.1 IC50 16
IVGTVZGLPHBTJV 8.1 IC50 16
KNUGHTXEXHMVQH 8.1 Ki 2
NICYKALLTQWBJN 8.1 Ki 2
ONFTYQQDJPXOLJ 8.1 Ki 2
QRZNWQBPKJMWHT 8.1 Kd 2
QVIQGNJPFOVZBZ 8.1 Ki 16
WGALJYRAUSZYPN 8.1 Ki 3
YHNNMZUUFMJQQY 8.1 IC50 16
AKFWDSCDLSTTJA 8.1 Ki 2
FIZTZZUELBWXAD 8.1 Ki 4
HGJUDXDUSGEVOX 8.1 Ki 6
WTCWMXBHKDJZDF 8.1 Ki 2
XQXFLYIUHYKDHV 8.1 Ki 4
DIAJWVOXHUCVAW 8.1 Ki 2
PPDJULIFZKACJD 8.1 Ki 2
PXCVVFWVLHUINV 8.1 Ki 5
XNNXOBKNOQSNCB 8.1 Ki 5
XRGYXMGEGDHNIO 8.1 Ki 2
ZONZZNQCOBYHOG 8.1 Ki 2
GSPMAICRXXSRDC 8.1 Ki 2
2D structure