Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
KLCFWSMDTGPJFU 8.3 Ki 2
WZNQGAWPCOPXOK 8.3 Ki 4
XUQGVVDGCDLCBJ 8.3 Ki 2
ZDWVXHPNJXPYJD 8.3 Ki 2
IREBWVNSEHBJRT 8.3 Ki 6
PQAZYCAWLLSXHO 8.3 Ki 6
QQKKCXYUPJTQBC 8.3 Ki 4
SQWDLBUOGWAKID 8.3 Ki 2
ZLLRNHZUVNVZMO 8.3 Ki 2
RHPXLQPYTRXEPL 8.3 Ki 2
XMMBCPSXQSTYKO 8.3 Ki 2
ZWWZTFYQCITUTK 8.3 IC50 16
BCOWBMDVBZPNTD 8.2 Ki 6
PXVVGKZGOHGYOO 8.2 Ki 2
ZLTZGADBISMZKB 8.2 Ki 4
ZMZBVSYTZFHKSN 8.2 Ki 2
ZFOFJXFVCJQXBL 8.2 Ki 3
BTLWEEGNXUJKKB 8.2 IC50 16
GXAQMBSYBNUQQZ 8.2 Ki 2
KIVQXKXZISOGBE 8.2 Ki 17
NHJRHDMRNNOSLV 8.2 Ki 5
NKIYALPHXLYICR 8.2 IC50 16
YIJHOBQVCMYCNA 8.2 Ki 5
YUSWMAULDXZHPY 8.2 Ki 20
ZRRVSALMQDOQAX 8.2 Ki 16
AUZCXFQYQQUAFH 8.2 Ki 7
BELGLGAAMPTDSH 8.2 Ki 2
UQOQENVWVOMXQR 8.2 Ki 2
YLPHFEFMBAMSKS 8.2 Ki 5
YOSWCJYMYAKWFV 8.2 Ki 2
BDISWVKOOATATE 8.2 Ki 16
GTOBFJHFOZIFFU 8.2 Ki 5
PAWVTIRLBCFWOI 8.2 Ki 2
JIDATJIBBMYJET 8.2 Ki 2
KCWCNDXYAPQOHU 8.2 Ki 5
MBBOXTKOOFAZLI 8.2 Ki 16
OYXXATFJACEJGE 8.2 Ki 6
AKFWDSCDLSTTJA 8.2 Ki 2
UKTUKCYHGVTZRH 8.2 Ki 2
BFDLKCJRLLXZFO 8.2 Ki 2
PKSKIVNMTHKBOS 8.2 Ki 2
QNLKJSGZMGMFBW 8.2 Ki 6
QORLMYYHZLDYOR 8.2 Ki 9
WDTGOYDHZIXMQO 8.2 Ki 7
YUOOYQDBXTWPKL 8.2 Ki 16
ZJQHPWUVQPJPQT 8.2 Ki 17
SJAGJFDQMIAULO 8.2 Ki 6
GQIVRYNNTCEOBX 8.2 Ki 8
KCWYSAXQZARGNH 8.2 Ki 2
OTQXKRRISJPTFS 8.2 IC50 16
2D structure