Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
DYSDYZCGZCYPCT 8.4 IC50 16
LMXUGQJMQSMLIQ 8.4 Ki 17
OSMYMXKHKOTLKC 8.4 Ki 7
UULFOYXSWNADTF 8.4 IC50 16
VXVLSQVFRWSMKF 8.4 Ki 6
VCPRTCGXKBSFJJ 8.4 Ki 4
YQYRRRVQWIMSFP 8.4 Ki 5
MKNXZRAKHYWDOS 8.4 IC50 16
QBYZDDIMNITMSB 8.4 Ki 6
VAJLZGPUVKNCRO 8.4 Ki 6
XQUJTESAXUTXNH 8.4 Ki 16
AYVAVBFBOCMUHW 8.4 Ki 6
INSVCYRFDCTMIA 8.4 IC50 5
ZPSBXQBYCQOCEU 8.4 Ki 6
CFMPKKXOXYNZHF 8.4 Ki 6
SOLFHEZOCDBPSQ 8.4 Ki 4
ZFVQZRCEZOITAU 8.4 Ki 2
FNEDDGRJWXWDNZ 8.3 IC50 5
HOXYFGSUNKVYSV 8.3 Ki 6
JTYYMOMTGZSRFM 8.3 IC50 16
PPLHNABOBXLAJU 8.3 Ki 4
WLHRDALLBOSVLX 8.3 Ki 6
IZOOOJDTIJXRIF 8.3 Ki 2
JTGPXCIJDIEQSX 8.3 Ki 4
NMIWQCPJXNFYRR 8.3 Ki 5
SNJUGZNPLIFITQ 8.3 Ki 2
BIBRQTYVULTGSH 8.3 Ki 4
JLERSVYBQKFVHN 8.3 Ki 2
IVVHFTRDYKTGCC 8.3 Ki 6
LTYUPBZLKIUGQX 8.3 Ki 8
YGKSPOBIXHTPMV 8.3 IC50 16
YNQYEEDREDAATO 8.3 Ki 2
KYEPYRBAELNJAO 8.3 Ki 2
ACMQMUZDLQDWTK 8.3 Ki 16
CBKOOGJFEQBENF 8.3 Ki 4
CLNVSRPCLJHOQX 8.3 Ki 2
CNFLHWVYIFARIM 8.3 Ki 7
DDLIGBOFAVUZHB 8.3 Ki 3
GOCZPCXRIJMRNR 8.3 Ki 16
JKDJAOQUTMBBQB 8.3 IC50 5
LPAODQAWVMEXKR 8.3 IC50 16
PHOATQSOBKATTD 8.3 Ki 16
PTRXPVDOTUGGHW 8.3 IC50 16
RAVIZVQZGXBOQO 8.3 Ki 3
RRMCHLUXWQTEQR 8.3 Ki 2
IAIZAMKHEDKXAK 8.3 Ki 6
XRRMKGIMNWBQJX 8.3 Ki 3
BKFSRIWWQZTOIW 8.3 Ki 5
DVKHCFDZNVGRQT 8.3 Ki 16
IVHDILBRMPOXID 8.3 Ki 2
2D structure