Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
PFSCOMOMUBXDBR 8.6 Ki 4
QZDWWRKBDPYMIP 8.6 Ki 6
WGRVAGIQTHEEQW 8.6 IC50 16
ACHPNNOYBNCORU 8.6 Ki 8
FNNPSIGQQWCKKB 8.6 Kd 5
CHIFCDOIPRCHCF 8.6 IC50 16
CHQPOBHNDRMXFK 8.6 Ki 18
KCEIOBKDDQAYCM 8.6 Ki 5
FUTRDVKMGNYUPP 8.5 Ki 6
HSKAYWQXMCMXAQ 8.5 Ki 3
KVKYGVOAHGNAKZ 8.5 IC50 17
LENHHZQGSWCZJW 8.5 Ki 16
LZTHAJBUMOQDLU 8.5 IC50 3
NXLVFWXJLBOCPO 8.5 Ki 2
RYLDZJANGRBUGW 8.5 IC50 16
RZXWKGHDRQNABH 8.5 IC50 4
UPPLJERIZONGME 8.5 Ki 6
OFBIFZUFASYYRE 8.5 Ki 16
FBBGZDOIPFFHLI 8.5 Ki 4
JXUDSFIVAUVTDY 8.5 Ki 2
VMKZXEMKFBINKN 8.5 Ki 3
LOZNAQDBHKVLRN 8.5 Ki 6
RZOFEWOHNOOHND 8.5 Ki 6
CUICGHSKDSXIRX 8.5 Ki 6
FLTICUPGYVYGAM 8.5 Ki 5
YWVNAIWRDXBOOS 8.5 Ki 6
ACUNYYFYYWOKOD 8.5 IC50 16
IBIAGNJTCFFVTB 8.5 Ki 5
LCQOTTUTLOUTNO 8.5 Ki 2
OJVFFZLXISLIFZ 8.5 Ki 6
UOYBEURVYWDNBS 8.5 Ki 5
ZGEGOFCLSWVVKG 8.5 Ki 5
MVBVNOZDVRVMNH 8.4 IC50 16
MZGKIGRVCYKVPS 8.4 Ki 6
OEIRQQZGARGKRG 8.4 Ki 6
OPOBFCRVBWVOQZ 8.4 Ki 2
OTWGFFXBGMUFBP 8.4 Ki 6
JYQBFIUGGKNLDH 8.4 Ki 6
LJRIFLWERUHAIZ 8.4 Ki 8
DSKYZAOKCWQIRI 8.4 Ki 4
IRYAGFJMRZLHGE 8.4 Ki 6
LSVOXYMZIGSSNB 8.4 Ki 6
NEOUOHDNZDRDNJ 8.4 IC50 16
OKGJPMZATLJSGV 8.4 Ki 6
PPTYJKAXVCCBDU 8.4 Ki 7
ZWWXXHQAJKCRDM 8.4 Ki 6
ALBKMJDFBZVHAK 8.4 Ki 16
AXPGZURVLRWNBR 8.4 Ki 16
BZVWONIGXAYZIT 8.4 IC50 16
CDWXZILKRXSANI 8.4 IC50 16
2D structure