Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
SRAWBNFSMIHBEM 8.9 Ki 8
VBXZLYYHFDVNEN 8.9 Ki 6
VWMUAQXLZGFQGW 8.8 Ki 2
YTGZSWOWFGVAFH 8.8 Ki 7
NTEUDQFHQWGEBH 8.8 Ki 5
QSEBFHRZNPGODU 8.8 Ki 6
BNQJKHFCSDKTCD 8.8 Ki 4
JAOIJSLHKQEWQB 8.8 Ki 4
PYXJKYJAFMLYMS 8.8 Ki 6
QAMUWRFOZKONDU 8.8 IC50 7
XJRDHPKTMGWJGN 8.8 Ki 6
ZBNZXTGUTAYRHI 8.8 IC50 102 Yes
QVOYXYWXOMVGNY 8.8 Ki 4
BQSIRVPTCKHWKR 8.8 Ki 5
IHDXFSAXAJRBOG 8.8 Ki 5
PHYVZWNIDCNYML 8.8 Ki 2
STHRYAZDXIDVJO 8.8 Ki 6
KBMIXEOSQPPORV 8.8 Ki 8
OJLYUGSSUKAWJC 8.8 Ki 16
PCKMQUISQMUBKK 8.8 Ki 4
UVTIJQDSGQQUDX 8.8 Ki 5
DNSPBVIIBSAYPW 8.7 Ki 5
KVKYGVOAHGNAKZ 8.7 IC50 16
WAPAOOACIDZLKD 8.7 Ki 8
NHJFEXZXSCFYRX 8.7 Ki 6
TXIWNLQFRATZFL 8.7 Ki 4
HJIQKECDKLWXGE 8.7 Kd 2
OLKUNPKISSHQBO 8.7 Ki 6
WIACWFSVQJVNGF 8.7 Ki 5
XBPAHSBPWSBJHT 8.7 Ki 6
YVTIEXKHDRKBSM 8.7 IC50 4
SHTOUNSWZVCSOU 8.7 Ki 16
QTEUJQNPMLXVLL 8.7 IC50 16
VJMXGRAYTDRKAO 8.7 Ki 6
ZDGLRCMEFVYZHG 8.7 Ki 6
AOZALWRGTMILIK 8.6 Ki 6
HOQUSTXYXSUJDG 8.6 Ki 6
AGXQLQJBYPTKJV 8.6 Ki 6
CHMFFBQMSYJXTP 8.6 Ki 6
CLMNGHYEDSVQIK 8.6 Ki 6
GWERFVJRQFKXQG 8.6 Ki 5
RWHXHODEPUBXTK 8.6 Ki 2
QIZPCEVRKTWHIE 8.6 IC50 16
GTLAYADJMQDCQJ 8.6 Ki 5
OXRXBJGSNZVEPW 8.6 Ki 4
AHHSTGLUTRNWRJ 8.6 Ki 6
QQJIGGMPLKYXPX 8.6 Ki 2
AWOOMIRCBITDFK 8.6 Ki 6
GXKGSEUULCEOTM 8.6 Ki 5
OKOKWNYOLUGIGN 8.6 Ki 3
2D structure