Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
RYIVVNHBYBYXHF 9.1 IC50 16
VZKRZUPJCVFVGR 9.1 IC50 16
FTBGMXWQYKNAKT 9.1 Ki 6
LLHQBHOWDZNCNK 9.1 Ki 5
RUOVJURXWIHZPL 9.1 Ki 5
QYSYOGCIDRANAR 9.1 Ki 7
FVFFDKKTXYVCCW 9.1 Ki 16
GFQMHVYMEKXHDT 9.1 Ki 6
AJWPZYMLAILYCO 9.1 Ki 5
BJYKRVMKNGJKKZ 9.1 Ki 6
LHGSGTVATLBNGO 9.1 Ki 3
NZMJFRXKGUCYNP 9.1 Ki 6
MNTGRSPARUFALM 9.1 Ki 5
YJZGQBGGTBIAOP 9.1 IC50 16
ZQLPLWRQUVVKJZ 9.1 Ki 6
KVTRKSLNWMZSSN 9.0 Ki 4
JYKXGGXAKPOFML 9.0 Ki 3
NPBFSLFGBCAWAF 9.0 Ki 6
AAFXZNIGLSLXPH 9.0 IC50 2
AQKFCEWRKDXGMK 9.0 Ki 16
IPHSQMSRIWZULE 9.0 Ki 16
IYYLIZWRYYVEPH 9.0 Ki 4
KDMMIKQMHNBKAV 9.0 Ki 17
KOVRZNUMIKACTB 9.0 Ki 17
PUNLHXOQDSEUQP 9.0 Ki 4
QCILNSKJADMOQI 9.0 Ki 4
RLFKILXOLJVUNF 9.0 Ki 16
UKHFPVCOXBJPIN 9.0 Ki 17
VJVAWKPXJCDEQG 9.0 IC50 16
XKDRJZMAMYYSIZ 9.0 Ki 2
DGBIGWXXNGSACT 9.0 Ki 16
PUZIHDVBQKJHLY 9.0 Ki 4
BSBLYLUAUVTSMM 9.0 IC50 16
LIFDPEORUVTOCP 9.0 IC50 4
OIVNHVRINWMDTH 9.0 Ki 5
PCEHLVFMKNNXOA 9.0 Ki 2
UFTKNTUWDMJOIX 9.0 Ki 16
ZAYUCIMDULREJZ 8.9 Ki 4
HNGRWUCKESPKRC 8.9 Ki 6
NURMFSYNABAOFU 8.9 Ki 6
OBQABQYFCKQGFL 8.9 Ki 3
PYEJACCXPZGJAH 8.9 Ki 2
QWWODAPIEHJFQG 8.9 Ki 16
VMDKDKVHHDTDAL 8.9 Ki 4
XGMPKZHPHLEVGE 8.9 Ki 4
XXRKXVKJMSIZSM 8.9 Ki 6
JOFWLTCLBGQGBO 8.9 Ki 8
JNJUWXAKLRKXII 8.9 Ki 6
KYKSBUKRCPZJCX 8.9 Ki 4
LWWWGLNBPILIGM 8.9 Ki 5
2D structure