Target Details
| UniProt AC | P14867 |
|---|---|
| Gene Symbol | GABRA1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit alpha-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 1,420
- Clinical molecules 3
- Avg pChEMBL 7.51
KEGG Pathways (8)
Associated Diseases (4)
Active Molecules (1,420)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OKZDZISQRKZKRC
|
6.0 | Ki | 2 | — | |
SZHSENNQOQSFEA
|
6.0 | IC50 | 16 | — | |
IUQSZUWRMNDZII
|
6.0 | Ki | 6 | — | |
GKHILVGVNGQMGS
|
6.0 | Ki | 2 | — | |
PHAFJLAQYPGVOC
|
6.0 | Ki | 2 | — | |
PHAFJLAQYPGVOC
|
6.0 | Ki | 2 | — | |
VCGRFBXVSFAGGA
|
6.0 | Ki | 6 | — | |
BARMYQHAEVRRFP
|
6.0 | Ki | 6 | — | |
BBQPVOQVHLCYFA
|
6.0 | Ki | 2 | — | |
DHLJRIFIBJGWBS
|
6.0 | IC50 | 16 | — | |
DQDLJDCSJFQOHI
|
6.0 | IC50 | 16 | — | |
GCTOZKWOFVUEAW
|
6.0 | IC50 | 16 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
IHFBPDAQLQOCBX
|
6.0 | Ki | 18 | — | |
KVZVPZYFPDOIMI
|
6.0 | IC50 | 16 | — | |
LOLNCKZNZWWETB
|
6.0 | Ki | 2 | — | |
MAVYALTWHWZSCK
|
6.0 | IC50 | 3 | — | |
RYFIWEJRWHTFBM
|
6.0 | IC50 | 16 | — | |
SOYRXCGRSSKEAM
|
6.0 | IC50 | 2 | — | |
ZOJGLIUFBPODLH
|
6.0 | Ki | 6 | — |