Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
CPWJDGKKDQPBKJ 6.1 Ki 2
FAHMQYRQDMWTRG 6.1 Ki 2
HYJUIJYNZHZBOK 6.1 IC50 16
INPWMTZRFFFMOA 6.1 Ki 2
NGYKELBMVXBFSM 6.1 Ki 5
PUMYFTJOWAJIKF 6.1 Ki 2
UPXSOIKTRIGNGR 6.1 Ki 6
WJEPRNMCEBRSDB 6.1 IC50 16
AFQKQBVQNAFSCA 6.1 Ki 2
KFJIZPKNMXRHEO 6.1 Ki 2
OXSWCVXEQZIBGE 6.1 IC50 3
WYEOFGFJCZYTHC 6.1 Ki 2
XDRLVLSTZNMYLB 6.1 Ki 2
YLZBNNDOEUIHFB 6.1 IC50 16
YTFLGZYWUGHFRL 6.1 Ki 2
ZMBXNSVOASWJOO 6.1 Ki 2
APPBGPRMFVUPRH 6.1 IC50 3
CXNUOOTVTMVRCI 6.1 IC50 3
FWZBUGMDRBQDHJ 6.1 Ki 6
LKUSWPRPRBXYPH 6.1 IC50 16
PQGDUNWRHHLMNT 6.1 IC50 9
SOYCFODXNRVBTI 6.1 Ki 6
VKMJGKFQKLVODR 6.1 IC50 16
VAEZVMCCCWEXEH 6.1 Ki 16
ZLQICIASTSXSFD 6.1 Ki 2
FUULVCWWUPGUMY 6.1 Ki 16
FVEJOOHXPUFGSK 6.1 Ki 2
QANMGLSLKPATOE 6.1 Ki 2
RGLUZPFSHJVPPP 6.1 Ki 2
UUZBPRCBLKYBQP 6.1 Ki 4
UYXLFIXVNVPFAS 6.1 Ki 2
DMFKLCONGDUSKT 6.1 Ki 2
IELTUHSCGWKNTD 6.1 Ki 2
IEXRFFQPFNOGAP 6.1 Ki 2
PIPOCLOMPZRSLC 6.1 Ki 4
ZXYMHGABHZSFOI 6.1 Ki 16
AKOKEYRHKIETQQ 6.1 Ki 2
DOOGDICMBOTQOZ 6.1 IC50 16
KGNWRICPWILABJ 6.1 Ki 6
RMMFOEVSBRAPQP 6.1 Ki 2
UYITUPHIEXJHKX 6.1 Ki 2
NEOJJVVOYKDEHZ 6.0 Ki 6
PJMYDDGWVUCELC 6.0 Ki 6
QCWSWDXAJBAYEA 6.0 Ki 2
SNUJIMQFPFCPCC 6.0 Ki 5
KDVOBKXBJSUGHB 6.0 Ki 2
PCGLDGXLCXIRGT 6.0 Ki 2
SLNCMJYPLFSUGO 6.0 Ki 16
XPTMQLMSBUSJOL 6.0 Ki 4
GBAKVEWPYUIGHN 6.0 Ki 2
2D structure