Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
BZIBRALMCDHACX 6.2 Ki 17
JWTQJUQJIRWZLA 6.2 Ki 16
ODWCGGCCGLKRAK 6.2 Ki 16
REIWWVZOVOIYMD 6.2 Ki 2
SFMVPQDIOHQZIK 6.2 Ki 2
XZTRSBKCRFMSHO 6.2 Ki 6
ZWNZTSDJEOGSPF 6.2 Ki 2
HVJGMCGDOFRWHL 6.2 Ki 5
NHXHETTUSFLPHY 6.2 Ki 2
TXPKEBVGMYWHJR 6.2 IC50 3
VDDATJOZLCYXHB 6.2 Ki 6
VTWITWDVHKQWCL 6.2 Ki 2
VYEPAZHUFFXYDH 6.2 Ki 6
ICRYUJPBYIPXQF 6.2 IC50 16
JIVGBDBCGKVLCY 6.2 Ki 6
UDAPJVKQJQNWQL 6.2 Ki 2
ZYTWOBRUUCLPMR 6.2 Ki 2
DQOWOBNQAJJKEH 6.2 Ki 2
LPOYLZZUEKLEBW 6.2 Ki 2
ZMKDYQONTIIETL 6.2 Ki 16
GDSKAAMFSMUYMJ 6.2 Ki 2
OJOTYQLMNVPQBO 6.2 Ki 16
RMBCZRNLGKJEAK 6.2 Ki 2
RRAXPPHKWFOGGL 6.2 Ki 16
WQIWYEISPHMPOA 6.2 IC50 16
YKVBFMDDXCMYHI 6.2 Ki 5
ARCJBXYEOMXBSZ 6.2 IC50 16
CTPREUOHTKHCHT 6.2 IC50 16
DPISUGVHZBSEIR 6.2 IC50 3
IZQOSQCYDUORJW 6.2 Ki 2
OJKALFLWJGRIRN 6.2 Ki 2
WOQHIJSDFJSXHI 6.2 Ki 2
XFUAEWGHLXLENC 6.2 IC50 16
BSEVRQDRIQMBCV 6.2 IC50 16
DHEXTYZLLGWEFS 6.2 Ki 16
DHZINDHXJITJQU 6.2 Ki 2
QUJXQESBGREUDF 6.2 Ki 2
VPHVDBRFNLXIHE 6.2 Ki 2
WEDYAXJXVWGXMB 6.2 Ki 6
XZUVYGZTGVSFPM 6.2 Ki 2
YEWWURAOECHIQL 6.2 Ki 2
HBOSSQBJUBOEJN 6.1 Ki 16
IDYXWWMDHPHNDU 6.1 Ki 2
KVMKDFFHDINSSZ 6.1 Ki 3
RKSUNQHPGFRQHL 6.1 Ki 6
RMFRINBLHMRFLI 6.1 Ki 6
ARMIIMXWCNOAOC 6.1 Ki 2
IADROWGKULIMIX 6.1 Ki 3
NAPZANZEQXWANH 6.1 Ki 2
XVFJUDUNNHPHLN 6.1 IC50 16
2D structure