Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
FNZFELZOBRBQJY 6.3 IC50 16
FYBWPCCAELGEHR 6.3 Ki 4
IATKEJBVROWZSN 6.3 Ki 2
IGCSLIVTBUKKRS 6.3 IC50 16
IVNZVVINRJLGRR 6.3 Ki 4
OWKXSFJRGOXMHI 6.3 Ki 2
SRJOCJYGOFTFLH 6.3 Ki 16
VFWOXQNFPHOBLO 6.3 IC50 3
YMDCFKGDSKTSDY 6.3 Ki 2
ZSWDNCJKCGDTKT 6.3 Ki 4
GAGMZQZBWNYDQU 6.3 Ki 6
JLLCYCAJCAQIHF 6.3 Ki 2
KFMFWOCTCNKUIB 6.3 Ki 6
KNJIPGCWYQXXPI 6.3 Ki 2
SZDYQTCZTLGXBX 6.3 Ki 6
YNMUMZXMMNJDIN 6.3 Ki 4
KMYUMBZLLVOGAP 6.3 Ki 2
LHDPGSHJSSZMRH 6.3 Ki 6
PZWMQJZDDYQYGN 6.3 Ki 16
YLZWVRAOJGXWTI 6.3 Ki 4
LFONXNFQWUEXIC 6.3 Ki 2
YDLSCFILSJHEPL 6.3 IC50 3
CFFHDCIRJSILAR 6.2 Ki 2
CMVRRVIUBQXVIK 6.2 Ki 2
CBBFXXVRQALAPG 6.2 Ki 2
FXIDXTIMKAEBGY 6.2 Ki 7
JDBPBOLDVHXIDJ 6.2 Ki 6
KGIVKXMZIJEMJQ 6.2 Ki 2
KUMNWRPRQLCGBZ 6.2 Ki 2
KUMNWRPRQLCGBZ 6.2 Ki 2
MWAUZLNCUAEKNR 6.2 IC50 2
NFYKGVIGVXLJTO 6.2 Ki 2
OGPGSYNCKSLJOF 6.2 IC50 2
ZEEOGWVZWOURAE 6.2 Ki 16
ZOEVKYRFHVGOOY 6.2 Ki 2
BTGRTTKTGRILMF 6.2 Ki 2
DAPYUYZNPMJDNB 6.2 Ki 2
SAVPBGVTWKUBOS 6.2 Ki 2
SRNKTNDYXGQRST 6.2 Ki 2
YOOKLJJRQNYLGH 6.2 Ki 2
ANTSCNMPPGJYLG 6.2 Ki 7
FCBLAIZVPBQHMO 6.2 Ki 2
FCKVAABCJRWYHI 6.2 Ki 2
HGXDYOKZLZBFJW 6.2 Ki 2
HSXSMQSDLMVYCV 6.2 Ki 2
NDRWXFUZQPBELD 6.2 IC50 3
NLCBGONMLZXCDS 6.2 Ki 2
NTKWVYCGMNXXNM 6.2 Ki 2
OMGOVFIKWLKTPS 6.2 Ki 16
QTZCODMFYAFKIE 6.2 Ki 2
2D structure