Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
NQFQEBQBZXSXIX 6.4 IC50 16
RBMPSWHARBABOC 6.4 Ki 6
UFSSPXFMMJZZDU 6.4 Ki 4
VNFZCRPFALLSNM 6.4 IC50 16
XOFGLRKYNSZCQZ 6.4 IC50 3
SQPWTARSPNZNEI 6.4 IC50 16
VIZDSLSEFNMSIJ 6.4 Ki 4
VSVKLTLXHHNTOE 6.4 Ki 4
KNURUKDSCWMMSN 6.4 Ki 2
QCSFXCHHKYXLHE 6.4 Ki 16
YFEZLTPSCJWVHI 6.4 Ki 16
KQQPWYMLATZBCF 6.4 Ki 2
LTSAESFXDBXRGS 6.4 Ki 3
YOJAHANNNITYMX 6.4 Ki 16
ZSDPALDTMGRNKW 6.4 Ki 2
CYGBAIOJMMSNSX 6.4 Ki 2
LEGPDWOWUFGLMP 6.4 Ki 3
PLDDKFUCCWRCBG 6.4 Ki 2
RXJAQIBDEJFUCL 6.4 Ki 6
YVIVUMAFAKNWHC 6.4 Ki 6
AEPFXRGRJZMVIF 6.3 Ki 17
MXUSCXPVOCAUMX 6.3 Ki 2
OJTLKYOKROEASR 6.3 Ki 4
QSOBDJYLKIXMJX 6.3 Ki 2
UIANKUAHFCTBLR 6.3 Ki 2
ZUUXQQXURVQFGG 6.3 Ki 3
BHJKLRZKDBSSKN 6.3 Ki 6
COFOXGPFFPFDIE 6.3 Ki 2
HCSPQICLTPISJP 6.3 Ki 2
IUVGMHPHSQSOGI 6.3 Ki 2
JBTLCAMUYYCXTA 6.3 IC50 16
LKTVCZVRYOFEAX 6.3 Ki 2
NSTKOSLZMSLHPO 6.3 Ki 3
BAGQLZQXEXAEAA 6.3 Ki 2
GCTGWUUTZLTQAR 6.3 Ki 6
LURVKJAOOMWPMR 6.3 Ki 2
NGYKELBMVXBFSM 6.3 Ki 5
VUKNNEXTWWCNCW 6.3 Ki 3
CQMLETFIENAKAA 6.3 IC50 2
HMRRNXHWVOACEA 6.3 IC50 3
LTIQJQOJEAIYPU 6.3 Ki 6
SGVYZSLDFHARFK 6.3 Ki 6
YCQFFXDKKZNVEE 6.3 Ki 6
ZXRVKCBLGJOCEE 6.3 Ki 5
BDGWCPYUERFMMY 6.3 Ki 16
NTKWVYCGMNXXNM 6.3 Ki 2
RQNGTQFJWSNXHS 6.3 Ki 2
UMYWGMKUCZAQJO 6.3 Ki 16
UVGSGGRQOUHBMK 6.3 Ki 6
ZLHFILGSQDJULK 6.3 IC50 37 Yes
2D structure