Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
KPKJEFIYLPVANT 6.5 Ki 4
HARMZUHRUKGCNG 6.5 Ki 8
HJGRBNHROFTASJ 6.5 IC50 16
LDSZEQFXAQLMOV 6.5 Ki 4
QCDKBYHARZQRIV 6.5 Ki 5
RAKFVWDVZYUQCI 6.5 Ki 2
YHZXFRGWTKYPKS 6.5 Ki 16
ZSEDMNMFODMQRD 6.5 Ki 5
GAQCKHAXURZXGX 6.5 IC50 16
HRCUSGLGVAUZHK 6.5 Ki 2
MHVBIDYSCZQVSY 6.5 Ki 5
SEUKIVWIQMZCJE 6.5 Ki 6
SZAYALFNNDVKGO 6.5 Ki 2
WORTYRSSHFTZAB 6.5 Ki 6
WRZBXBIKXIYAGJ 6.5 Ki 6
PMDUNHOOULGNCQ 6.5 Ki 6
QWZAWUIUHQADCS 6.5 Ki 2
VEWLYIAEUXDQBW 6.5 IC50 16
ARLPBUKOJFUUPW 6.5 Ki 2
GDVGLPNNOCDLLD 6.5 IC50 16
DLCURRAFWAXUPF 6.5 Ki 5
HHFBDROWDBDFBR 6.5 IC50 40 Yes
UDBOMYAYEKMWDV 6.5 Ki 4
WDMOSRJVOUIQMD 6.5 Ki 3
GEFDSAOHFGLQEZ 6.5 Ki 17
WCTCMHZWHMFZFN 6.5 Ki 17
DDSULWHSYUPHBK 6.5 IC50 16
KHVVJKLNKLQLJZ 6.5 Ki 288
VRIQRWQZIAEDLB 6.5 Ki 2
ZLAPTIDQRXJQQL 6.5 Ki 16
XRWYYMUIIXMQBL 6.5 IC50 16
OCZOXZDVTVVPSN 6.4 Ki 2
VHUKNSIDUVPWBR 6.4 Ki 2
CPBKEZZAUBJVEY 6.4 Ki 2
FICZDYQNTMRYOG 6.4 Ki 2
IZUFYFBJMFQQAV 6.4 Ki 2
LXQGNWWMMCBHEW 6.4 Ki 2
MAHFVAHPQSLLJF 6.4 Ki 288
QUBHUQVCFZIJRF 6.4 Ki 3
CVZIRDLTVVTXNF 6.4 Ki 6
DAYQXLQRTQODQF 6.4 Ki 16
DNCFKDLZZSXXJP 6.4 IC50 16
GDQHTINQBXUUJK 6.4 Ki 4
ISEATUPRORNMRO 6.4 Ki 2
MPIBCTUFGUTVSG 6.4 IC50 3
QHJVRBLRBSIYGE 6.4 Ki 4
UDARHNNVNUUUEB 6.4 Ki 2
UGPCGLRXJCIGIY 6.4 Ki 2
ZMGVJHPLOILGKH 6.4 Ki 2
MUPIUJYENVWEKT 6.4 IC50 16
2D structure