Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
MZUQNVRYMWOVSR 6.7 Ki 6
NSEGTDJUUQGMNZ 6.7 Ki 3
PGTVWKLGGCQMBR 6.7 IC50 16
QKZNNAUSAVZXNE 6.7 Ki 16
GRHSJPRDKRVXDK 6.7 Ki 6
HGPFVUUTSFNGNR 6.7 Ki 18
GSJSXDQXHDAYLZ 6.7 Ki 6
ISYJVUADIFBVQO 6.7 Ki 2
LIIRYFLHPZDMEC 6.7 Ki 6
BBSNJCBFCWNPBH 6.7 Ki 8
NGWYCOVARFKQDW 6.7 Ki 9
ZHNHRBPYLNHOJB 6.7 Kd 2
AAZYXOJZFFSUBA 6.7 Ki 6
GMVMGIYPRPPNMB 6.7 Ki 16
PUJKPXPABLQPRA 6.7 Ki 3
UDLTUJYBFNCMJX 6.7 Ki 7
UDLTUJYBFNCMJX 6.7 Kd 2
XDUPLYSGJVWGTM 6.7 Ki 5
ZRKQHHNVLRRZFQ 6.7 Ki 16
DEPRZKLICJNMGM 6.7 Ki 3
PTRPQDMPYNOBTR 6.7 IC50 16
UDTZRZLWBNBNCX 6.7 Ki 2
DATCQVJMADOCRS 6.7 IC50 16
GFJMSLRUMDAFSY 6.7 Ki 6
GXUSNZYZTBJMIT 6.7 Ki 16
NSVRIDBPWFCPNQ 6.7 Ki 6
WKMUEHICTZESCZ 6.7 IC50 3
ZGEMNNHBINYTKL 6.7 IC50 3
SINAJPKUKOSXOT 6.7 IC50 16
XHWVFLWDNDWXHW 6.7 Ki 2
IPXNFQNXWOFDQD 6.7 Ki 6
KDOQEEMQPHIANX 6.7 Ki 2
MPASHPJAIUOWCK 6.7 Ki 9
OOTAQHRUCFIGFZ 6.7 Ki 7
SYYSMZCCSNLTHZ 6.7 Ki 2
WFRRJMYHDPXXFB 6.7 Ki 16
YWCLXVVWMQVKRF 6.7 IC50 16
ABTNVOCRBNFBHY 6.6 Ki 2
CELFESKDAXZKDL 6.6 IC50 16
HXXGVDKGNHCARX 6.6 IC50 16
ILFYWHUZKNCDEU 6.6 Ki 6
INIXNNKFVDXPBJ 6.6 Ki 3
KUZLDKPQBCXMLJ 6.6 Ki 6
LDPMPCNDVKFVIW 6.6 Ki 6
NRCNHRJESVKFJO 6.6 Ki 6
BNANSHHVRHDWHQ 6.6 Ki 2
NESUAJPAOMXMJC 6.6 Ki 6
VMNYVCMDPUOQEL 6.6 Ki 16
ACVGNKYJVGNLIL 6.6 IC50 16
ARBXYFIBGCCVTN 6.6 IC50 2
2D structure