Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
LQKOTGTWBANJBS 6.8 Ki 6
KTFRBKXLNKKPEA 6.8 IC50 16
UIEAPAOHCIQRQL 6.8 Ki 6
XHXRMYICRMVHBK 6.8 Ki 4
ANKFABXSPKCYOQ 6.8 Ki 6
DGWAMRKYNYINRJ 6.8 IC50 16
DXCKAYBKZBTPNN 6.8 Ki 6
GTRFGCMGMHCDPF 6.8 Ki 8
QQXJSYFEJVOQLZ 6.8 IC50 16
UQXPONWWSBAXMI 6.8 IC50 2
VDMSNGMYNVTHDD 6.8 IC50 3
VGZQARXDBOOWBF 6.8 Ki 16
AWLPAJABQMKXOE 6.8 Ki 3
HICZHPFZMDTJBP 6.8 Ki 5
LOFKMRMDVCEZEF 6.8 Ki 7
DSTVUBPAEXKNMB 6.8 Ki 6
FVLVVJPWTSTRCM 6.8 Ki 6
JTQDBIFZWJTIIQ 6.8 Ki 16
JXKAURVNHHPPND 6.8 IC50 16
MXTPRZSAMHVJFI 6.8 IC50 2
OFFQUPKDTOZERU 6.8 Ki 6
PRGDQIDWABTGRF 6.8 Ki 4
QMCOPDWHWYSJSA 6.8 Ki 2
QTEBXBALJGPXEP 6.8 Ki 3
RHARCGZTSJROQQ 6.8 Ki 16
RLKPTPBBRCFHEK 6.8 IC50 16
RXBGGFMEZUKQME 6.8 Ki 2
XMLLCLHYZOZSEG 6.8 Ki 6
ZLMXJIGMRPRGMM 6.8 Ki 6
BPKZCNBWMWKTIB 6.8 Ki 4
BXKSCEUJEPDZBI 6.8 Ki 16
OWAIKGZBRPVIGC 6.8 Ki 2
STQWWORVIGBLOE 6.8 Ki 16
VGKZDCNKIZAJPG 6.8 Ki 2
XAXZXMJZHNVJEQ 6.8 Ki 16
IYEJMUDDGFBLEF 6.8 Ki 6
VFWOXQNFPHOBLO 6.8 IC50 3
CGOOGLSJSVATGZ 6.8 Ki 16
FLHRNVLCKMTQAP 6.8 Ki 17
JQHJWKNJYLNAFL 6.8 IC50 16
UKXDLKBYAPSHDL 6.8 Ki 6
VSVSOYLJDWHVLX 6.8 IC50 3
AFJRYPJIKHMNGL 6.8 Ki 6
HLRBYKMPMSUTAX 6.8 Ki 6
KYAAEHKCLYGUJO 6.8 Ki 6
WDBDNAQYXVEMIT 6.8 Ki 6
XLKFCRQJPWBJNW 6.8 IC50 16
KPKJEFIYLPVANT 6.8 Ki 4
CGVJPQYHXQIFPE 6.7 Ki 16
MAMCCEALLBBOGS 6.7 Ki 6
2D structure