Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
FQDQLHDSVITISC 7.0 IC50 16
NVRZICQXMRMPGV 7.0 Ki 2
YEFFWDGMWBFKHL 7.0 Ki 16
ZYQKNGNVEVNORP 7.0 Ki 6
RMGFIVKKLZZKNY 7.0 IC50 16
XVRONCOEBFKZEW 7.0 IC50 16
BULOMLIWEVCBPE 6.9 Ki 6
FTLMOIDJQCYEHM 6.9 Ki 2
NMMJOCVBNVTBNP 6.9 Ki 16
GQXSRHIFUJLCSW 6.9 Ki 16
JYXHNHBKWZQGLB 6.9 Ki 16
BSJXQBNOVPYHPA 6.9 Ki 6
GZGLGVQROXSNSN 6.9 Ki 9
HWOWPGLTTSFLOQ 6.9 Ki 16
LCCYGVBXMXVHRW 6.9 Kd 2
LFKVDZOBBXOFEW 6.9 Ki 2
MJTBJNQOWBQCJE 6.9 Ki 2
PRAPAJSGMGWZLK 6.9 Ki 3
VFKHADGYGKHTDK 6.9 IC50 16
LHSWKUZVAZKLHJ 6.9 IC50 16
NLHGXPUKOAOTRO 6.9 Ki 4
VFPUCBWBLOQFPU 6.9 IC50 16
XBJMMUWKPCJOBK 6.9 Ki 2
JXCPQLHXZUWOCZ 6.9 Ki 4
YZBJLGYBBNTKKL 6.9 IC50 16
CBAXLHGEEASOPH 6.9 Ki 6
QAXDJUNLAJMPAE 6.9 Ki 6
VXWQZPBYJRRNSX 6.9 Ki 3
VYRDWGGXTHOMJX 6.9 Ki 6
VHBFFQKBGNRLFZ 6.9 Ki 21
PVBWXOPKUUTANH 6.9 Ki 6
ACPUCHLYONVNTK 6.9 Ki 16
VMDUABMKBUKKPG 6.9 Ki 16
XCZACYJBBMAUSL 6.9 Ki 3
XYLGLGFZLQRDKD 6.9 Ki 16
BIHMYZHWJAFHBO 6.8 IC50 16
CAIDJZOHDFNJOZ 6.8 Ki 4
CEEIIGPEJDLELP 6.8 Ki 6
GZFUZKBKBLJQLQ 6.8 Ki 3
HOXKKBLQXUBSEI 6.8 Ki 6
INGJMHPGMVUEKY 6.8 Ki 6
JQLSECBWDAKQJE 6.8 Ki 6
KOTFZRCPKVQWPP 6.8 Ki 16
OWTXLWRGHNAFHX 6.8 Ki 6
PWDALQSYHZMANN 6.8 Ki 3
QUZHRQSFJYFDCO 6.8 Ki 6
SHHPYNVQBLHDPA 6.8 Ki 6
VJXWQJKLMZXRCW 6.8 Ki 6
XLKFCRQJPWBJNW 6.8 IC50 16
ZQWZTGULGCIKLX 6.8 Ki 6
2D structure