Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
HLKYSQGBIIIQJN 9.4 Ki 5
OGBTVLIUFUJHTH 9.4 Ki 5
GSLDBWNPXFIQAV 9.4 Ki 2
LICVBNQRZFPUHS 9.4 Ki 4
BGOCUVAKPSPUAI 9.3 Ki 2
QCNXINIQJHEAHO 9.3 Ki 4
WDCRWMNKRWOGOP 9.3 Ki 4
XKENJWNGLCKOBP 9.3 IC50 16
JLCBYDSLJHLQQB 9.3 Ki 5
NJUMMJUUDUYSKB 9.3 IC50 16
WRXDVVALWQGPMW 9.3 Ki 16
BGVDDMWFMIAGGF 9.3 Ki 5
BUTCFAZTKZDYCN 9.3 Ki 6
IPBXYXQZSUGQTK 9.3 Ki 5
KYDURMHFWXCKMW 9.3 Ki 6
NVETZYIXXYETLA 9.3 Ki 6
NVWCZRPXYVDQEE 9.3 Ki 5
DHWTVCHLMXAWGK 9.3 Ki 3
UWXAQZGCSSYTJL 9.3 Ki 6
FNCCIRFBYGUBRQ 9.3 Ki 5
SEWXZWMBVGJJPG 9.3 Ki 7
ULMLVGYYGWVNSC 9.3 Ki 3
BPTASZCHRIMWEF 9.3 Ki 6
IUHKSTINHDUYRO 9.3 IC50 16
MTNLFTKJHWYWQV 9.2 Ki 4
BLJPKQXXDFIIFR 9.2 IC50 16
IQKMZIHHJYCEKH 9.2 Ki 5
XJMIBNLJFYSGAR 9.2 IC50 16
ZKVGHURGXXUFQB 9.2 Ki 6
MTOXGGJOEHOEJT 9.2 Ki 5
XPSAGIQSESMIJK 9.2 Ki 6
VYBPWFTWAKMZPZ 9.2 Ki 5
BKIXSCDBYYIHQI 9.2 Ki 5
BWWQXKSOWUMHAQ 9.2 Ki 6
PFJHXYJLEIZLGQ 9.2 Ki 6
VSZZYAJBIGSJJF 9.2 Ki 4
KVQKVRWATUWLAO 9.2 Ki 5
NTQIDFIQUNKLIH 9.2 Ki 5
UPMDLTAPSSWEPU 9.2 Ki 4
LWUDDYHYYNNIQI 9.1 Ki 6
PCZLQMGFNUNVOM 9.1 Ki 6
PWFUHHSGSJDKCU 9.1 Ki 16
YLDRVNNGBACDSD 9.1 Ki 6
LHMYCKKRCBXCBI 9.1 Ki 5
BQDUNOMMYOKHEP 9.1 Ki 6
CJBGLZXUYDUSDI 9.1 Ki 2
CVOASAXXOXOGQG 9.1 Ki 5
ILFZZMYJRPZIPF 9.1 Ki 5
JFGUJXZLJIUVPZ 9.1 IC50 16
LYFROTHEKIFZAU 9.1 IC50 16
2D structure