Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
PRUQRKPURHYKRP 7.2 Ki 16
SOCJQMROXJKCQV 7.2 IC50 2
VAVBWHIBLOPOEM 7.2 Ki 16
IOOGUHXPDYRXFJ 7.2 IC50 16
XQPLNBUVGTUPTK 7.2 Ki 2
YMIKAQYPFQWUEM 7.2 Ki 7
IINVUOUPVKEBFS 7.2 Ki 5
NDFKYGUTDGWIHX 7.2 Ki 6
PTWRSNCLLAFDMD 7.2 Ki 3
UHSSVTHYXUDPRY 7.2 Ki 2
WCYJVRQPVHPWLQ 7.2 Ki 16
WHEUGJHMVJCNEP 7.2 IC50 16
XSXHDMUABOGLFX 7.2 IC50 2
NZBYBIYUIBGUGN 7.2 Ki 2
SINAJPKUKOSXOT 7.2 IC50 16
FUKXWTBJKBFICR 7.2 Ki 2
HRJQUDZTLASEPW 7.2 Ki 6
LMWOXZHQXIIVQI 7.2 Ki 3
LPOZDKMXSPAATL 7.2 Ki 16
MAZZBGKHYOJFSH 7.2 Ki 6
XXVQXGKSBMSCHX 7.2 Ki 6
KDGMRQJYYKGVCJ 7.1 Ki 7
QCQSTOYKSWTFNN 7.1 Ki 6
RDMWWTOMSYTLOT 7.1 Ki 6
VVCKCOBSJPEUNF 7.1 Ki 2
GMFUIVLIESEUHZ 7.1 Ki 6
KXZCHKGJBKPUPX 7.1 Ki 2
NFINWJGHOWQVKC 7.1 IC50 2
VOZOMZWSLGQRKP 7.1 IC50 16
YTBQKFMHGZGVAG 7.1 Ki 2
ZQZXBWMDLMNNQJ 7.1 Ki 2
DXRFLGVWSRQJHG 7.1 Ki 2
FESCSZDQOFYRDR 7.1 Ki 7
FNTHJTUPRVAXFZ 7.1 IC50 17
HWWJCYIYBBEGDP 7.1 Ki 6
LRKIZSIATCYGSA 7.1 Ki 3
OIKCREAGTIJWOO 7.1 Ki 6
YBRXFNLNMSTVNQ 7.1 IC50 16
BALGGUJCACDSLM 7.1 Ki 6
KZSDRHSSHPIBAO 7.1 Ki 6
NJHDFBWEGMPSBV 7.1 Ki 6
YINBZIQMPAZHMF 7.1 Ki 6
CAJUSRIHDIZNNF 7.1 Ki 6
DZCUZLPTNNFSNM 7.1 Ki 2
HRTSOMLTEJFUCO 7.1 IC50 16
KJMYFGDZNNIFLG 7.1 Ki 6
PGTVWKLGGCQMBR 7.1 IC50 16
AKDSPRXIQQMVKS 7.1 Ki 6
FHTNSYDGFUAOSS 7.1 Ki 2
FHXDHVUQGGBLGD 7.1 Ki 4
2D structure