Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
HMQQCASSOWMONY 7.4 Ki 2
ONIHNTIPKYMTGW 7.4 Ki 3
QMHTYKLXSOQULX 7.4 Ki 16
AVPMETBBKHOJBE 7.4 Ki 2
BXTBYBNRHFJYSX 7.4 Ki 2
CDRADZRGYBTOKU 7.4 Ki 6
CMUJABAHLCISIQ 7.4 Ki 6
DUZTVXKYJROMJJ 7.4 IC50 16
BMIKDIWICOAHJN 7.4 Ki 16
MSFAMEBSEKIVDI 7.4 Ki 16
VUZAUNZSDCMUTH 7.4 Ki 16
MRBNIDFDWVVALT 7.3 Ki 5
SAIRVAYGVLKBIG 7.3 Ki 6
ZZTJJGWSKYVZIG 7.3 Ki 6
HWUMRCHENDXGOC 7.3 Ki 2
LPKBUGHEXSSVCI 7.3 Ki 6
RAHUQMWUVSMABB 7.3 IC50 2
UXRDTECAKSYGRM 7.3 Ki 2
GWCQPEHFUKZODL 7.3 Ki 16
JSEPJHYIUICRFD 7.3 Ki 2
ACVGNKYJVGNLIL 7.3 Ki 5
GLOOEDBOHDKUMM 7.3 Ki 4
IADVCSUFBXJTCE 7.3 Ki 3
HEGJYRQUDMITRQ 7.3 Ki 6
NRJWKUBEWAELQW 7.3 Ki 2
NUXNKKUXSDGYTN 7.3 Ki 7
RHPSRJBQHFLHNQ 7.3 Ki 5
VBEASATUUNKOCC 7.3 Ki 2
VXDPUKHUSNJVCJ 7.3 Ki 6
YKYOQIXTECBVBB 7.3 Ki 7
BRTAZTLXPXQATA 7.3 Ki 2
GBBSUAFBMRNDJC 7.3 Ki 6
GWZLKOYBOFFDEB 7.3 Ki 6
NEECFEXLNIDWFK 7.3 Ki 2
QYEIQYJLVREYBI 7.3 IC50 16
RMPSDPZBGHYHQZ 7.3 IC50 2
SIBRGSBVGDWJAF 7.3 IC50 16
WGDPTKIWQGBNLZ 7.3 Ki 2
WHGIBMIKSVYLCR 7.3 IC50 16
YIIKQLCKNDAHHQ 7.3 Ki 8
YNGRKYAIISTAOT 7.3 IC50 2
AURFZBICLPNKBZ 7.3 IC50 16
NLKUQHZVJJAJEG 7.3 Ki 2
QRENCFPTMQNJCY 7.3 Ki 2
VOZJTMRCZHINKT 7.3 Ki 2
DGZYPGWWTKGBQP 7.3 Ki 16
FAZVYCLIQCGGCB 7.3 Ki 2
IPEQYLWHCRAOTC 7.3 Ki 6
KBFYDAGNYWSKLZ 7.3 Ki 6
LAKKZRKOENZKBW 7.3 Ki 2
2D structure