Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
HSUCRXNJMPDNOG 7.6 IC50 16
JNWDOTPNEZYWGO 7.6 Ki 16
NFMFVESVKLVYJR 7.6 Ki 7
QSBFNERLQPXCDQ 7.6 Ki 5
SQAIVYWNBGRPKS 7.6 Ki 2
UEBDAHFOLOMMDI 7.6 Ki 4
YBHLQPIYKPUFSS 7.6 Ki 6
ZPQLCRIOLZPVJB 7.6 Ki 6
FLTOAJWVMNMXMX 7.6 Ki 6
ISJKPUWGGXLQCI 7.6 Ki 5
JAFQEKAQGSQGTM 7.6 Ki 16
KQTMWRZAVOUNCI 7.6 IC50 16
VIEKPLVJCPXIIB 7.6 IC50 16
XLKKKDPUVUIHEL 7.6 IC50 16
YICWHQNQWIQUMG 7.6 Ki 5
YTUMMZANIYQNOM 7.6 Ki 8
ZDLKXIOQJJRYCW 7.6 Ki 6
KLKHVLINJXRNBG 7.6 IC50 4
LXRITECWUGVGTD 7.6 IC50 6
DLEZDQQOGQGPDX 7.5 Ki 6
LUDMNXOOXWWZDU 7.5 Ki 7
MMWKMKRWCPKFRA 7.5 Ki 6
QOICRVBHAUSMFA 7.5 Ki 6
RNQUVXLJHSQSIT 7.5 Ki 2
RTRHXDLGBINMNM 7.5 IC50 5
WDTNKNNGHGOKBH 7.5 Ki 9
YDLSCFILSJHEPL 7.5 IC50 3
YZRXMMCBUVDBFF 7.5 Ki 6
ZOCSXAVNDGMNBV 7.5 IC50 16
HAHDKXDDOBLEEH 7.5 Ki 3
PAGIUELYHAPFIM 7.5 Ki 2
SSJXJXJUHUAOQL 7.5 Ki 6
WOAZIFSEQSOHDW 7.5 Ki 2
XQDOFXHMSFUKQI 7.5 Ki 2
AANJEGNNNSDLGW 7.5 Ki 16
HBBBENORIXSUJV 7.5 Ki 6
LJXDYPITZRPEJE 7.5 Ki 2
MFHJVQXEYIWUCI 7.5 Ki 5
WPJDKKSDGLIQQB 7.5 Ki 16
XJCSIGHRPMXCCH 7.5 Ki 5
YGDRYLWBXSSWNT 7.5 Ki 2
ZXMSJXJLGNNGQW 7.5 Ki 2
ASUXILMTDDVWPD 7.5 Ki 7
BGETVQMBBYHJJF 7.5 Ki 6
CVNPFPRAINQAHI 7.5 Ki 5
DRCGHGOPCPUYAI 7.5 IC50 16
NKIYALPHXLYICR 7.5 IC50 16
OPLLZAJXBSDWMS 7.5 Ki 2
ZACQJMKEQBFUDN 7.5 Ki 6
BPPPQWRMTWGDJW 7.5 Ki 6
2D structure