Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
RMIQCBAOSNZENR 7.7 Ki 2
RSEMKXACIMVTQP 7.7 Ki 16
TUWKJMRKBCKTBU 7.7 Ki 2
ZRZOZCBSSVQEGD 7.7 Ki 6
WRDHNUVAWMYMJK 7.7 IC50 16
AURFZBICLPNKBZ 7.7 IC50 16
DXPCEAZKJSYFJM 7.7 Ki 6
IRDWCVIRNKWGSM 7.7 Ki 3
LTTJOUHFUIFFNF 7.7 Ki 2
MVCCGUFWBDSIHW 7.7 Ki 3
RBWPBJRIJOEHCN 7.7 Ki 6
RFYCGFKOGLYZKJ 7.7 Ki 6
ZFLBRINMIQTFNB 7.7 Ki 18
CJYPUCKDMBCYEH 7.6 IC50 16
GSQMITXEUGIGFD 7.6 Ki 3
JOHKRJNYKDHTID 7.6 Ki 6
LNPSYDJGQQETLB 7.6 Ki 16
RMIQCBAOSNZENR 7.6 Ki 2
TWQDMCPDTPVCQP 7.6 IC50 16
VHQCVUYEMJHQEX 7.6 Ki 16
VXYGMPPNCYIPDT 7.6 Ki 2
XQPLNBUVGTUPTK 7.6 Ki 2
BHXXVBIFJUPLTC 7.6 Ki 2
JHDNCJGODWCHES 7.6 IC50 16
LIXHLXZPUZQKCT 7.6 IC50 16
PDOZRVXKPBQAJH 7.6 IC50 16
QAMANTJYKWSLNP 7.6 Ki 6
RGDHMJMNRYQXCW 7.6 Ki 6
UHEYIOPHTBWBQN 7.6 IC50 3
BTCRVOSPHNKQGJ 7.6 Ki 6
JWLCOGXPTWMMDY 7.6 Ki 16
NCNYJRNYAGZTRG 7.6 Ki 2
GXYIMPYRUIKXIS 7.6 Ki 6
KBVJZOBCOIANOX 7.6 Ki 16
KJUPZRXGDNYFQT 7.6 Ki 6
KOMBGWPXIHBMLL 7.6 IC50 16
KWHWSXISOMCUPZ 7.6 Ki 16
LSHLIINFMYHQMQ 7.6 Ki 6
OSHQANHMWJQRHB 7.6 Ki 16
QUDSZGFPDUXASR 7.6 Ki 4
RDYMFSUJUZBWLH 7.6 IC50 6
SMJGKUZFWMGZEJ 7.6 Ki 2
ULMKSNRBNFFOJQ 7.6 Ki 16
ZSMNMYCBVFAPQG 7.6 Ki 6
ZWJGDMSWCKASII 7.6 IC50 16
FDUYIOSVUSYEQJ 7.6 Ki 6
KGRNGTYKNLBEPP 7.6 Ki 2
TUSMRQUKQRMRRW 7.6 Ki 2
ACZCJTHHWMBFKC 7.6 Ki 2
BXTBYBNRHFJYSX 7.6 Ki 2
2D structure