Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
YJQPSUGEFJEJIN 7.8 Ki 6
AHTXTFPELOVMKB 7.8 Ki 6
HOMGIOZFYSJYAP 7.8 Ki 2
KFRCPAXRUYFZQC 7.8 Ki 2
MQWOHTJLMXPEIA 7.8 Ki 2
NLEQOPYBIKKOPK 7.8 Ki 7
OVFRNPXWYQUNHR 7.8 Ki 4
RPWZDMRYJDLFFQ 7.8 Ki 2
TZEWBPGVTYPITP 7.8 IC50 5
YJYRFBZSNPRHKU 7.8 IC50 16
FVIWEOUHYRAQKY 7.7 Ki 6
GSPMAICRXXSRDC 7.7 Ki 2
HRNSOLSYHZMSCD 7.7 Ki 6
IBPJOIOGTFGBRO 7.7 Ki 6
PMFGUFKMTACZHR 7.7 Ki 6
RTHSDLLYNWWMSZ 7.7 Ki 6
WXCRCHQGSPOSLF 7.7 Ki 3
XDEHJKJHEDWFEK 7.7 Ki 2
BIVWQDOYGGWQHQ 7.7 Ki 2
PFKQLDDYRDGULP 7.7 Ki 2
QBWJMTOHSYOPBE 7.7 Ki 7
QJBCFALTTSBEEO 7.7 Ki 6
RJNFLJNUEOERRU 7.7 Ki 6
SNVZCVVNVLIROS 7.7 Ki 6
UIPGLQFPZVUUQW 7.7 Ki 16
VQENDYBPFSSMNH 7.7 IC50 16
YRHWMEGQCCRQAT 7.7 Ki 2
ZDWVXHPNJXPYJD 7.7 Ki 2
ZGZMACKWWYQZLH 7.7 Ki 2
DUUKVMKDBTYKFQ 7.7 Ki 3
KDOQEEMQPHIANX 7.7 Ki 2
SDMRVWKQZCYVGP 7.7 Ki 2
VREFGVBLTWBCJP 7.7 Ki 7
XGCMWZQFAAILJM 7.7 Ki 2
BYEKIJACVDAPTD 7.7 Ki 16
FJADGXRCKLHLAK 7.7 Ki 3
HCJVWLPVQMYLOI 7.7 Ki 8
LLAKESJIQFAQJA 7.7 IC50 16
NSYQRTSKIVJYPU 7.7 Ki 2
QILRYFCEXLFIDS 7.7 Ki 7
ZQLRGKFMMVAALA 7.7 Ki 2
HMQQCASSOWMONY 7.7 Ki 2
RYODDIOYGKHDCF 7.7 Kd 2
AZIRFKLEFANUIC 7.7 Ki 6
BOEVLQCJGHTZLQ 7.7 Ki 2
FQDQLHDSVITISC 7.7 IC50 16
HKLYPSSDHPAOJM 7.7 IC50 16
IEDCFFRFAIAYGF 7.7 Ki 7
IKXSFQFVTQDDAR 7.7 Ki 6
MLRKAMHWRLRODO 7.7 Ki 4
2D structure