Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
RBMPSWHARBABOC 7.8 Ki 6
WAEXHEOACCAOSS 7.8 Ki 16
GAONFNHSQRTFJA 7.8 Ki 6
HXSMEVAYWUOWMI 7.8 Ki 2
HYMHVNNHIASECU 7.8 IC50 5
RDVZJHHFIHQSMW 7.8 Ki 2
RQCRZVPWNJSJSP 7.8 Ki 6
VLFMZVVYNJAVLQ 7.8 Ki 2
GMTZLHADUFDDDN 7.8 IC50 5
LAGQGYLPSNORIA 7.8 Ki 2
MNIOVVAGLOIPRL 7.8 Ki 2
IMMPJABTWMVMPJ 7.8 Ki 16
IQXJMMLNUIUGIQ 7.8 Ki 16
PNRLOCDAUHBIHX 7.8 IC50 16
ULDBOWIRGDMZPF 7.8 Ki 8
VSHQZNAELPBUKM 7.8 Ki 2
VVBYXJYBLBPAEN 7.8 Ki 6
XMPCGSSQTOZYPB 7.8 Ki 5
AAMAQVCMQYBDCZ 7.8 Ki 5
AUNROIIKFNFPRC 7.8 Ki 2
MVHGYSDYQMHHMG 7.8 Ki 2
WLJWRZRVPBWFBZ 7.8 Ki 2
ZHLQLUZELIBEJT 7.8 Ki 2
CKZVPJOTELQSHC 7.8 IC50 16
DRCWBQAOFNLXIV 7.8 Ki 7
DZPQKPSHACGLKC 7.8 Ki 6
FVYRQIQXAYUADB 7.8 Ki 2
OOAXMNBBGAIJCT 7.8 Ki 7
PCRRXYJDKILUID 7.8 Ki 6
QCHBQARHFYCDNV 7.8 IC50 16
RJOMRLSAWXNFSU 7.8 Ki 4
YOGKDBMNVNETRZ 7.8 Ki 6
ZFPVOBQMGRHOBJ 7.8 IC50 16
GKHLLLCEUXLULG 7.8 Ki 2
JKCPXTTYNRGYQQ 7.8 Ki 4
OWGSYSGRQRUUDH 7.8 Ki 2
ZYJJWEOKCFKOTD 7.8 Ki 2
CLNVSRPCLJHOQX 7.8 Ki 2
LGUQZQBSKOYXKY 7.8 Ki 2
AYRJXCIMSHQLPG 7.8 Ki 6
HJNOESUOZGNLKO 7.8 Ki 6
HRNSOLSYHZMSCD 7.8 Ki 5
JWZNKJCEYMWLHS 7.8 IC50 16
MEWGBPFYMUBENF 7.8 IC50 16
NAXZRUMPHRMRDF 7.8 IC50 16
NRPDDGBNDOXOCO 7.8 Ki 2
UYPWOMKFYXODIW 7.8 Ki 7
VXOXRIDQOBACKW 7.8 Ki 16
XNIDSAVZEZPOBT 7.8 Ki 6
XUJMJGTVTZESCM 7.8 Ki 7
2D structure