Target Details
UniProt ACP14867
Gene SymbolGABRA1
Protein NameGamma-aminobutyric acid receptor subunit alpha-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,420
  • Clinical molecules 3
  • Avg pChEMBL 7.51
Top Co-occurrence Targets
Active Molecules (1,420)
InChIKey pChEMBL Type Targets Clinical
CGMJQQJSWIRRRL 10.3 Ki 6
LCDOZBPYZHDFGO 10.0 Ki 5
LTRYPGNCHZSXSI 9.9 Ki 3
NAGYYVWENUNCDU 9.9 Ki 3
TUYGGVAJDAZCIC 9.9 Ki 3
FYOXWZFDOADHOW 9.8 Ki 6
KKWDMTXJUXKNOU 9.8 Ki 7
KKXPFXBGMGQSMA 9.8 Ki 3
QXZGSQAJHBQSSV 9.8 Ki 4
MZFKWSFOAVBLQM 9.8 IC50 16
WDBBCFFNOHDOBT 9.8 Ki 5
AJTIJRUGVRMRDN 9.8 Ki 5
LDXAQEAQNGTFAB 9.7 Ki 4
PTTQXDBPTFOCMT 9.7 Ki 6
VJCYGDVWTVTYGY 9.7 Ki 2
FIXFKUDATBTRAZ 9.7 Ki 4
WFPXOWCKXUEKCA 9.7 IC50 16
YIGPWWJHDOXRHC 9.7 Ki 4
YMMRGIIZANFGIG 9.7 Ki 6
DLGWSCNXWHDMHZ 9.7 Ki 4
GOIFCXRIFSYPFG 9.7 Ki 5
BYMDBFGHCDTBMT 9.7 IC50 16
VACJUKKURQMWHE 9.6 Ki 5
ISZRIZPRXUQOMU 9.6 Ki 5
KVKWRJDNIJTMGN 9.6 IC50 16
BCLNCXBDWXPRAH 9.6 Ki 4
ZRKDDZBVSZLOFS 9.6 Ki 6
QKIWQBLNTSQOLY 9.6 Ki 6
WQYYZNGOTUCWQX 9.6 Ki 5
RYKBQSSZEXHGJL 9.6 Ki 5
GTPDUXMCZZEOBE 9.5 Ki 4
RWUOGVWORJUNJA 9.5 Ki 4
WMBPDZBHEAETLZ 9.5 Ki 3
KMGQMDWTLIZLHG 9.5 Ki 4
QIWRIQRYIRGJCG 9.5 Ki 4
VQOOIUSVMMFXEJ 9.5 Ki 4
LWUDDYHYYNNIQI 9.5 Ki 7
AZLLXOVNVMQRNP 9.4 Ki 4
CUCYVGNNTAIIAN 9.4 Ki 4
CMSKDYKEKYIJSD 9.4 Ki 5
FAEJWVCMADNLAQ 9.4 Ki 4
MPEKCHDBHNYAJG 9.4 Ki 2
RXMRVZANJZUNED 9.4 Ki 3
GMDXFYPWVIKBFF 9.4 Ki 4
PEBWTLIJBCZFOA 9.4 Ki 6
RKXGEVUMNLOCDX 9.4 Ki 3
BCEWAHBYIZQWJY 9.4 Ki 5
BFKIZTLCAFUHPD 9.4 Ki 2
PWTUVRWHZWTHMS 9.4 Ki 2
QUUNMICPMYIHFS 9.4 IC50 16
2D structure