Target Details
| UniProt AC | P14756 |
|---|---|
| Gene Symbol | lasB |
| Protein Name | Elastase |
| Organism | Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22644 / CIP 104116 / JCM 14847 / LMG 12228 / 1C / PRS 101 / PAO1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07504 (FTP) PF03413 (PepSY) PF01447 (Peptidase_M4) PF02868 (Peptidase_M4_C) |
Summary
- Multi-target molecules 2
- Clinical molecules 1
- Avg pChEMBL 6.82
Active Molecules (2)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZPHBZEQOLSRPAK
|
7.2 | Ki | 5 | — | |
IIOCRGOBAHXAAI
|
6.4 | IC50 | 4 | Yes |