Target Details
| UniProt AC | P14618 |
|---|---|
| Gene Symbol | PKM |
| Protein Name | Pyruvate kinase PKM |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00224 (PK) PF02887 (PK_C) |
Summary
- Multi-target molecules 4
- Clinical molecules 1
- Avg pChEMBL 6.59
KEGG Pathways (10)
Active Molecules (4)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QFJCIRLUMZQUOT
|
7.3 | IC50 | 9 | — | |
MWKSRKSEWLRPBL
|
6.8 | Kd | 1075 | — | |
FSWBAMMIGFKJBV
|
6.3 | IC50 | 6 | — | |
KZNIFHPLKGYRTM
|
6.0 | IC50 | 21 | Yes |