Target Details
| UniProt AC | P14616 |
|---|---|
| Gene Symbol | INSRR |
| Protein Name | Insulin receptor-related protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00757 (Furin-like) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 17
- Clinical molecules 7
- Avg pChEMBL 6.94
KEGG Pathways (2)
Active Molecules (17)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
8.2 | Kd | 231 | Yes | |
HZTYDQRUAWIZRE
|
8.1 | Kd | 40 | Yes | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
XZXHXSATPCNXJR
|
7.7 | Kd | 165 | Yes | |
AILRADAXUVEEIR
|
7.3 | IC50 | 75 | — | |
LQVXSNNAFNGRAH
|
7.3 | Kd | 33 | Yes | |
CXQHYVUVSFXTMY
|
7.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.3 | Kd | 149 | — | |
PKCDDUHJAFVJJB
|
7.1 | IC50 | 13 | — | |
GCIKSSRWRFVXBI
|
6.5 | Kd | 109 | Yes | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
MOSKATHMXWSZTQ
|
6.3 | IC50 | 16 | Yes | |
KTEIFNKAUNYNJU
|
6.2 | Kd | 114 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |