Target Details
| UniProt AC | P14598 |
|---|---|
| Gene Symbol | NCF1 |
| Protein Name | Neutrophil cytosol factor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16621 (NCF1_PBR_AIR) PF08944 (p47_phox_C) PF00787 (PX) PF00018 (SH3_1) |
Summary
- Multi-target molecules 5
- Clinical molecules 1
- Avg pChEMBL 7.1
KEGG Pathways (12)
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Fc gamma R-mediated phagocytosis
- Fluid shear stress and atherosclerosis
- Leishmaniasis
- Leukocyte transendothelial migration
- Lipid and atherosclerosis
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- Phagosome
- Prion disease
Associated Diseases (2)
Active Molecules (5)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RKEWSXXUOLRFBX
|
8.6 | Ki | 5 | — | |
RAPZEAPATHNIPO
|
7.7 | Ki | 28 | Yes | |
DYEFUKCXAQOFHX
|
6.4 | IC50 | 31 | — | |
KZEUBCUXBNEMSQ
|
6.4 | IC50 | 2 | — | |
RBTBFTRPCNLSDE
|
6.4 | IC50 | 5 | — |