Target Details
| UniProt AC | P14091 |
|---|---|
| Gene Symbol | CTSE |
| Protein Name | Cathepsin E |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07966 (A1_Propeptide) PF00026 (Asp) |
Summary
- Multi-target molecules 66
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (1)
Active Molecules (66)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SXQPECMJHHMDFO
|
10.0 | Ki | 5 | — | |
ICOVQVRWYNMTQP
|
9.4 | IC50 | 2 | — | |
GCZHKZTYTMTFGU
|
9.4 | IC50 | 3 | — | |
FAXGPCHRFPCXOO
|
9.3 | IC50 | 14 | — | |
BDYFZQDNIIZQQW
|
9.3 | Ki | 5 | — | |
MQDDTALXSBQTQP
|
9.3 | Ki | 5 | — | |
NXDIWJUYMKBICN
|
9.1 | IC50 | 3 | — | |
JZYWSTGTBRHGTL
|
9.1 | IC50 | 5 | Yes | |
OCAGLXMEXWSQMK
|
8.7 | IC50 | 3 | — | |
DVRJOUXWYVOMLR
|
8.7 | Ki | 5 | — | |
HZWNNIVRFLRAQW
|
8.7 | Ki | 4 | — | |
ZKQFFTQZNAYNHR
|
8.7 | Ki | 4 | — | |
YZCWZTFSJLJQLC
|
8.5 | Ki | 4 | — | |
ACLGFPBLVWSDHZ
|
8.5 | Ki | 5 | — | |
YZORPUYWQSMGBV
|
8.5 | Ki | 4 | — | |
DLWWAEZPTACWPK
|
8.4 | IC50 | 3 | — | |
VOLBHADFPHYYLF
|
8.3 | IC50 | 2 | — | |
GZHSLBYVXGDJDF
|
8.3 | Ki | 4 | — | |
OFVXANJIRQGPPI
|
8.3 | IC50 | 2 | — | |
ULGBSRGDBHJMRG
|
8.3 | IC50 | 3 | — | |
TVDHOONBSNHWKJ
|
8.1 | IC50 | 3 | — | |
MRUQYXTWPXNCJI
|
8.1 | IC50 | 2 | — | |
YZORPUYWQSMGBV
|
8.0 | Ki | 4 | — | |
SQKBSPJLGLPLAW
|
7.9 | IC50 | 3 | — | |
UFJYUSGISGEOOF
|
7.8 | Ki | 3 | — | |
YTIOGZLHYJDYTK
|
7.8 | Ki | 5 | — | |
PVHMTQKFPXCDJQ
|
7.7 | Ki | 3 | — | |
VZRWUYQWJBSEAG
|
7.7 | IC50 | 3 | — | |
CJLWKFUIIJXJBZ
|
7.6 | IC50 | 3 | — | |
GOSHIBGNLKXPDZ
|
7.6 | IC50 | 2 | — | |
YDCNYSQITCUGST
|
7.6 | Ki | 4 | — | |
GJTOCPGDDLTBBD
|
7.5 | IC50 | 3 | — | |
XKXGRRZAMDHVGR
|
7.5 | Ki | 4 | — | |
BYPTUSJUZLWKPS
|
7.4 | IC50 | 3 | — | |
WFMVRFNXMBGKEW
|
7.4 | IC50 | 3 | — | |
GNXRLNXFKDAFQU
|
7.4 | Ki | 4 | — | |
VIIORGGCTLITHW
|
7.3 | Ki | 5 | — | |
UXROPHBUPUPWOI
|
7.3 | IC50 | 3 | — | |
LRAVCRYIDZOXGD
|
7.3 | IC50 | 2 | — | |
KQBGZTOQVQFMJZ
|
7.2 | IC50 | 3 | — | |
WFMVRFNXMBGKEW
|
7.2 | IC50 | 3 | — | |
JAZOCUNZCUBRJX
|
7.1 | IC50 | 4 | — | |
BAGQHZIZGKYGNB
|
7.1 | IC50 | 2 | — | |
CQQMWBPWYUPVOC
|
7.1 | Ki | 4 | — | |
SHXBHHDCBHQKLF
|
7.0 | Ki | 4 | — | |
PSNGTIQWNUJCAN
|
7.0 | IC50 | 6 | — | |
QGUDJRLYHSLQDK
|
7.0 | IC50 | 2 | — | |
AKZOFLGCSPMBPS
|
7.0 | IC50 | 3 | — | |
CZXLJTCMHQXVJW
|
7.0 | IC50 | 2 | — | |
KJQYIOYOHBXLEG
|
6.9 | IC50 | 4 | — |